1. Membrane Transporter/Ion Channel
  2. Potassium Channel

VU0529331 

目录号: HY-112705
产品使用指南

VU0529331 是一种适度选择性的不含 GIRK1 的 G蛋白门控内向整流钾 (non-GIRK1/X) 通道抑制剂,在 HEK293 细胞中,对 GIRK2 和 GIRK1/2 的 EC50 值分别为 5.1 µM 和 5.2 µM,同时对 GIRK4 同源通道也有作用。

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VU0529331 Chemical Structure

VU0529331 Chemical Structure

CAS No. : 1286725-49-2

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Description

VU0529331 is a modestly selective non-GIRK1-containing G protein-gated, inwardly-rectifying, potassium channel (non-GIRK1/X) activator, with EC50s of 5.1 µM and 5.2 µM for GIRK2 and GIRK1/2 in HEK293 cells, respectively, also effective on GIRK4 homomeric channel[1].

IC50 & Target

EC50: 5.1 µM (GIRK2), 5.2 µM (GIRK1/2)[1]

References
Molecular Weight

384.43

Formula

C₂₂H₂₀N₆O

CAS No.

1286725-49-2

SMILES

O=C(C1=NC=CN=C1)N2CC3=C(N4C=CC=C4)N(C5=CC(C)=C(C)C=C5)N=C3C2

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Shipping

Room temperature in continental US; may vary elsewhere

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The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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产品名称:
VU0529331
目录号:
HY-112705
需求量:

VU0529331

Cat. No.: HY-112705