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(R)-BAY1238097 

目录号: HY-112316A
产品使用指南

(R)-BAY1238097 是BAY1238097 的低活性 R 型异构体。BAY1238097 是一种有效的、BET与组蛋白 结合的选择性抑制剂,通过下调c-Myc水平及下游转录组,在AML (急性髓性白血病) 和MM (多发性骨髓瘤) 模型中表现出较强的抗增殖活性。

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(R)-BAY1238097 Chemical Structure

(R)-BAY1238097 Chemical Structure

CAS No. : 1564269-85-7

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Size Price Stock Quantity
10 mM * 1 mL in DMSO ¥2750 In-stock
5 mg ¥2500 In-stock
10 mg ¥3900 In-stock
50 mg ¥12500 In-stock
100 mg ¥21000 In-stock
200 mg   Get quote  
500 mg   Get quote  

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Description

(R)-BAY1238097 is the R-isomer with lower activity of BAY1238097. BAY1238097 is a potent and selective inhibitor of BET binding to histones and has strong anti-proliferative activity in different AML (acute myeloid leukemia) and MM (multiple myeloma) models through down-regulation of c-Myc levels and its downstream transcriptome[1][2].

IC50 & Target

BET[1].

References
Molecular Weight

451.56

Formula

C₂₅H₃₃N₅O₃

CAS No.

1564269-85-7

SMILES

O=C(N1N=C(C2=CC=C(N3CCN(C)CC3)C=C2)C4=CC(OC)=C(OC)C=C4C[C@H]1C)NC

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Shipping

Room temperature in continental US; may vary elsewhere

  • 摩尔计算器

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The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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产品名称:
(R)-BAY1238097
目录号:
HY-112316A
需求量:

(R)-BAY1238097

Cat. No.: HY-112316A