2. GPCR/G Protein Neuronal Signaling
  3. Adrenergic Receptor
  4. α2C adrenoceptor agonist 1

α2C adrenoceptor agonist 1 (Compound A) 是一种具有口服活性、高选择性和非中枢神经系统穿透的 α2C-肾上腺素受体激动剂，EC50 和 Ki 值分别为 108 nM 和 12 nM。α2C adrenoceptor agonist 1 可以用于鼻塞的研究。

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α2C adrenoceptor agonist 1 Chemical Structure

α2C adrenoceptor agonist 1 Chemical Structure

CAS No. : 928115-79-1

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α2C adrenoceptor agonist 1 相关抗体

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查看 Adrenergic Receptor 亚型特异性产品:

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α adrenergic receptor β adrenergic receptor

  • 生物活性

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生物活性

α2C adrenoceptor agonist 1 (Compound A) is an orally active, highly selective, and non-central nervous system penetrating agonist for the α2C-adrenoceptor, with EC50 and Ki values of 108 nM and 12 nM, respectively. α2C adrenoceptor agonist 1 can be used in the study of nasal congestion[1].

IC50 & Target

Alpha-2C adrenergic receptor

108 nM (EC50)

Alpha-2C adrenergic receptor

12 nM (Ki)

体内研究
(In Vivo)

α2C adrenoceptor agonist 1 (Compound A) (5 mg/kg; p.o.; 单剂量) 在 Sprague-Dawley 大鼠中的脑渗透性较差，其平均 Cmax、Tmax 和曲线下面积值分别为 0.8 μM、0.7 h和2 μM•h[1]。

MCE has not independently confirmed the accuracy of these methods. They are for reference only.
分子量

315.37

Formula

C16H21N5O2
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

α2C adrenoceptor agonist 1 相关分类

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  • Do most proteins show cross-species activity?

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Keywords:

α2C adrenoceptor agonist 1928115-79-1Adrenergic ReceptorBeta Receptornasal congestionInhibitorinhibitorinhibit

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