2. GPCR/G Protein
  3. Free Fatty Acid Receptor
  4. GPR40 agonist 5

GPR40 agonist 5 (化合物 I-14) 是一种口服有效的 GPR40 (G 蛋白偶联受体 40) 激动剂，其 EC50 值为 47 nM。GPR40 agonist 5 可降低血糖水平，改善糖耐量。GPR40 agonist 5 对 2 型糖尿病小鼠的高血糖状态有充足的控制作用。

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GPR40 agonist 5 Chemical Structure

GPR40 agonist 5 Chemical Structure

CAS No. : 2443384-60-7

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GPR40 agonist 5 相关抗体

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生物活性

GPR40 agonist 5 (compound I-14) is an orally active and potent GPR40 (G protein coupled receptor 40) agonist, with an EC50 of 47 nM. GPR40 agonist 5 decreases the levels of blood glucose and improves the glucose tolerance. GPR40 agonist 5 has sufficient effectiveness for the control of hyperglycemia state in type 2 diabetic mice[1]. GPR40 agonist 5 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.

IC50 & Target

EC50: 47 ± 9.8 nM (GPR40)[1]
分子量

440.49

Formula

C27H24N2O4
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

GPR40 agonist 5 相关分类

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

GPR40 agonist 52443384-60-7Free Fatty Acid ReceptorFFARType 2 diabetes mellitusT2DMFree fatty acid receptor 1FFA1G protein coupled receptorGPR40 agonistsPhenylpropanoic acidHepatotoxicityInhibitorinhibitorinhibit

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