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  2. Androgen Receptor
  3. PF-06260414

PF-06260414 

目录号: HY-108326
产品使用指南

PF-06260414 是具有口服活性的、非甾醇的选择性雄激素受体调节剂 (SARM)。

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PF-06260414 Chemical Structure

PF-06260414 Chemical Structure

CAS No. : 1612755-71-1

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Description

PF-06260414 is an orally active and nonsteroidal selective androgen receptor modulator (SARM)[1].

In Vitro

PF06260414 has potent AR agonist activity in a cellbased transcriptional reporter assay, with a concentration of a drug that gives half-maximal response of approximately 0.3 nM (79% efficacy vs DHT)[1].

In Vivo

PF-06260414 has fast absorption (median Tmax, approximately 1–2 hours), a mean t1/2 of approximately 6.9 to 12.8 hours, time-independent PK properties and dose proportionality[1].

Molecular Weight

302.35

Formula

C₁₄H₁₄N₄O₂S

CAS No.

1612755-71-1

SMILES

N#CC1=NC=CC2=C1C=CC(N(C[C@H](C)CN3)S3(=O)=O)=C2

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Keywords:

PF-06260414PF06260414PF 06260414Androgen ReceptorInhibitorinhibitorinhibit

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产品名称:
PF-06260414
目录号:
HY-108326
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