1. Membrane Transporter/Ion Channel
  2. Calcium Channel

Calcium Channel

Calcium channel is an ion channel which displays selective permeability to calcium ions. It is sometimes synonymous as voltage-dependent calcium channel, although there are also ligand-gated calcium channels. Voltage-gated calcium (CaV) channels catalyse rapid, highly selective influx of Ca2+ into cells despite a 70-fold higher extracellular concentration of Na+. Some calcium channel blockers have the added benefit of slowing your heart rate, which can further reduce blood pressure, relieve chest pain (angina) and control an irregular heartbeat.

Calcium Channel 相关产品 (103):

Cat. No. Product Name Effect Purity
  • HY-A0064
    Verapamil hydrochloride Antagonist 99.97%
    Verapamil hydrochloride 是一种 L 型钙离子通道 (calcium channel) 拮抗剂。
  • HY-B0470
    Neomycin sulfate Inhibitor >98.0%
    Neomycin sulfate 是一种氨基糖苷类抗生素,同时也是钙离子通道的阻滞剂。
  • HY-B0284
    Nifedipine Antagonist
    Nifedipine 是有效的钙离子通道 (calcium channel) 阻滞剂,常用于治疗心肌功能不全。
  • HY-B0282
    Acetylcholine chloride Activator >98.0%
  • HY-15553A
    Mibefradil dihydrochloride Inhibitor >98.0%
    Mibefradil dihydrochloride 是一种钙离子通道 (calcium channel) 抑制剂,选择性作用于 T 型 Ca2+通道,作用于 T 型和 L 型通道,IC50 分别为 2.7 μM 和 18.6 μM。
  • HY-B0768A
    Lomerizine dihydrochloride Antagonist 99.97%
    Lomerizine dihydrochloride 是一种双重的 L- 和 T 型电压门控钙通道 (calcium channel) 拮抗剂。
  • HY-13764
    Tetrandrine Inhibitor 99.49%
    Tetrandrine 是一种双苯基异喹啉生物碱,抑制电压门控钙离子通道 (ICa) 和 Ca2+ 激活的钾离子通道。
  • HY-103315
    Bepridil hydrochloride Antagonist 99.76%
    Bepridil hydrochloride 是一种钙离子通道 (calcium channel) 抑制剂,具有抗心绞痛的作用。
  • HY-B0265
    Nimodipine Inhibitor 99.87%
  • HY-15124
    Bay-K-8644 ((S)-(-)-) Agonist 98.34%
    Bay-K-8644 (S)-(-)- 是 L 型钙离子通道激动剂。Bay-K-8644 (R)-(+)- 激活 Ba2+电流 (IBa),EC50 为 32 nM。
  • HY-12542A
    Dantrolene sodium hemiheptahydrate Inhibitor >98.0%
    Dantrolene钠盐水合物是一种钙通道蛋白抑制剂, 抑制钙离子从肌浆释放, Dantrolene钠盐水合物是一种骨骼肌松弛药。
  • HY-B0106
    Levetiracetam Inhibitor
    Levetiracetam(UCB L059)是一种抗癫痫化合物。
  • HY-14656
    Diltiazem hydrochloride Antagonist 98.39%
    Diltiazem hydrochloride是钙离子流入抑制剂(缓慢通道阻断剂或钙拮抗剂)。
  • HY-19721
    ABT-639 Inhibitor 99.15%
    ABT-639 是一种新型选择性的 T 型 Ca2+ 通道阻滞剂。
  • HY-15125
    Bay-K-8644 ((R)-(+)-) Inhibitor 98.90%
    Bay-K-8644 (R)-(+)- 是钙离子通道抑制剂。Bay-K-8644 (R)-(+)- 抑制 Ba2+电流 (IBa),IC50 为 975 nM。
  • HY-B0233
    Isradipine Inhibitor 99.24%
  • HY-B0320A
    Cromolyn sodium Inhibitor 99.97%
  • HY-B0317B
    Amlodipine besylate Antagonist 98.21%
  • HY-17404
    Cilnidipine Inhibitor 99.92%
  • HY-12515A
    Nicardipine Hydrochloride Inhibitor 99.85%
    尼卡地平(Nicardipine; YC-93)盐酸盐是一种钙通道拮抗剂,已被广泛应用于控制的严重高血压等疾病,缺血性中风,脑外伤,脑出血等。
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