2. GPCR/G Protein
  3. GHSR
  4. GHSR-1a agonist-1

GHSR-1a agonist-1 (Compound 4b) 是一种具有口服活性的人源生长激素促分泌素受体 1a (GHSR-1a) 的激动剂，EC50 为 0.49 nM。GHSR-1a agonist-1 通过激活 GHSR-1a 来有效刺激内源性生长激素释放。低至 0.1 mg/kg 剂量的 GHSR-1a agonist-1 (口服) 即可增加 4 周龄大鼠体重和体长。GHSR-1a agonist-1 可用于儿童生长发育迟缓领域的研究。

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GHSR-1a agonist-1 Chemical Structure

GHSR-1a agonist-1 Chemical Structure

CAS No. : 3060887-25-1

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GHSR-1a agonist-1 相关抗体

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GHSR1a

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

GHSR-1a agonist-1 (Compound 4b) is an orally active agonist of the human growth hormone secretagogue receptor 1a (GHSR-1a), with an EC50 of 0.49 nM. GHSR-1a agonist-1 can effectively stimulate the release of endogenous growth hormone by activating GHSR-1a. GHSR-1a agonist-1 administered orally at a dose as low as 0.1 mg/kg can increase the body weight and body length of 4-week-old rats. GHSR-1a agonist-1 can be used in the research field of growth and development retardation in children[1].

IC50 & Target

GHSR1a

0.49 nM (IC50)

分子量

531.65

Formula

C30H37N5O4
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

GHSR-1a agonist-1 相关分类

  • 摩尔计算器

  • 稀释计算器

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

GHSR-1a agonist-13060887-25-1GHSRGrowth hormone secretagogue receptorGhrelin receptorInhibitorinhibitorinhibit

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