1. Metabolic Enzyme/Protease
  2. Phosphodiesterase (PDE)
  3. PDM-042

PDM-042 是一种有效的、选择性的、具有口服活性的磷酸二酯酶 10A (PDE10A) 抑制剂。PDM-042 对人和大鼠 PDE10A 显示出有效的抑制活性,IC50 值小于 1 nM,对其他磷酸二酯酶的选择性超过 1000 倍。 PDM-042可用于精神分裂症的研究。

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PDM-042 Chemical Structure

PDM-042 Chemical Structure

CAS No. : 1404488-48-7

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  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

PDM-042 is a potent, selective, and orally active phosphodiesterase 10A (PDE10A) inhibitor. PDM-042 shows potent inhibitory activities for human and rat PDE10A with IC50 values of less than 1 nM and more than 1000-fold selectivity against other phosphodiesterases. PDM-042 can be used for the research of schizophrenia[1].

IC50 & Target

IC50: <1 nM (for human and rat PDE10A)[1]

分子量

406.48

Formula

C21H26N8O

CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.

纯度 & 产品资料
参考文献
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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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PDM-042
目录号:
HY-160111
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