1. Signaling Pathways
  2. Metabolic Enzyme/Protease
  3. Drug Metabolite

Drug Metabolite

Drug metabolite results when a drug is metabolized into a modified form which continues to produce effects. Drug metabolism redox reactions such as heteroatom dealkylations, hydroxylations, heteroatom oxygenations, reductions, and dehydrogenations can yield active metabolites, and in rare cases even conjugation reactions can yield an active metabolite.

Drug Metabolite 相关产品 (28):

Cat. No. Product Name Effect Purity
  • HY-17366
    Clozapine N-oxide 99.98%
    Clozapine N-oxide (CNO) 是抗精神病药物氯氮平的主要代谢产物。 Clozapine N-oxide是 DREADD 系统的激动剂。
  • HY-13318
    Oseltamivir acid 98.60%
    Oseltamivir acid,是GS 4071的乙酯前药,是流感病毒神经氨酸酶的抑制剂,IC50 约为100 nM。
  • HY-100599
    Urolithin A 98.06%
    Urolithin A是具有抗氧化和抗增殖作用的鞣花酸的肠代谢物; 抑制T24和Caco-2细胞的生长的IC50值分别为43.9和49 μM。
  • HY-101406
    Thyroxine sulfate >98.0%
    Thyroxine sulfate是甲状腺激素代谢物。
  • HY-101107
    Allopregnanolone >98.0%
  • HY-G0002A
    Lurasidone metabolite 14326 hydrochloride Chemical 98.76%
    Lurasidone metabolite 14326 (hydrochloride) 是一种非典型抗精神病药物 Lurasidone 的活性代谢物。
  • HY-G0014B
    Quetiapine sulfoxide hydrochloride
    Quetiapine sulfoxide hydrochloride (Quetiapine S-oxide hydrochloride) 是 Quetiapinem 的主要代谢产物。Quetiapinem 是第二代抗精神病药。
  • HY-100645
    Trimethoprim 3-oxide >98.0%
    Trimethoprim 3-oxide 为一种三甲氧苄二氨嘧啶的初级代谢物。
  • HY-12772
    Hydroxy Itraconazole 99.60%
    Hydroxy Itraconazole 是 Itraconazole (ITZ) 的活性代谢物,Itraconazole 是一种三唑类抗真菌剂。
  • HY-B1398
    Ampyrone 98.86%
    Ampyrone 是一种试剂,在过氧化物酶与苯酚存在时,用于葡萄糖测定。
  • HY-101397
    Allopurinol riboside 99.04%
    Allopurinol riboside是别嘌呤醇的代谢物,能有效地抑制寄生虫。
  • HY-G0006
    Omeprazole metabolite Omeprazole sulfide 99.91%
    Omeprazole sulfide是Omeprazole的代谢物。
  • HY-G0014
    Quetiapine sulfoxide
    Quetiapine sulfoxide (Quetiapine S-oxide) 是 Quetiapinem 的主要代谢产物。Quetiapinem 是第二代抗精神病药。
  • HY-G0014A
    Quetiapine sulfoxide dihydrochloride >98.0%
    Quetiapine sulfoxide dihydrochloride (Quetiapine S-oxide dihydrochloride) 是 Quetiapinem 的主要代谢产物。Quetiapinem 是第二代抗精神病药。
  • HY-101407
    Nicotinamide N-oxide 99.45%
    Nicotinamide N-oxide是生物体内烟酰胺分解代谢物, 是高效选择性的CXCR2受体拮抗剂。
  • HY-G0011S
    Netupitant N-oxide D6
    Netupitant N-oxide D6是Netupitant N-oxide的氘代化合物标准品。
  • HY-G0011
    Netupitant metabolite Netupitant N-oxide
    Netupitant N-oxide是Netupitant的代谢物。
  • HY-G0007
    Omeprazole metabolite Omeprazole sulfone
    Omeprazole sulfone是Omeprazole的代谢物。
  • HY-G0010S
    N-desmethyl Netupitant D6
    N-desmethyl Netupitant D6是N-desmethyl Netupitant的氘代化合物标准品。
  • HY-15793A
    Trans (2,3)-Dihydrotetrabenazine
    Trans (2,3)-Dihydrotetrabenazine, 是抗精神病药物Tetrabenazine的体内代谢物,能够抑制囊泡单胺转运体 2 (VMAT2)
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