1. Signaling Pathways
  2. Membrane Transporter/Ion Channel
  3. SGLT
  4. SGLT Inhibitors

SGLT Inhibitors

SGLT1

SGLT2

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SGLT Inhibitors
Product Name SGLT1 SGLT2 Purity
Empagliflozin  
SGLT2
99.90%
Dapagliflozin  
SGLT2
99.97%
Canagliflozin  
SGLT2
99.70%
Phloretin
SGLT1
SGLT2
99.92%
Sotagliflozin
SGLT1
SGLT2
99.89%
SGLT1/2-IN-8
SGLT1
SGLT2
rel-Licogliflozin
SGLT1
SGLT2
Phlorizin
SGLT1
SGLT2
99.93%
Ipragliflozin
mSGLT1, IC50: 1380 nM
hSGLT1, IC50: 1876 nM
rSGLT1, IC50: 1166 nM
rSGLT2, IC50: 6.73 nM
mSGLT2, IC50: 5.64 nM
hSGLT2, IC50: 7.38 nM
99.71%
Ertugliflozin  
SGLT2
99.92%
Mizagliflozin
SGLT1
  99.20%
Dapagliflozin ((2S)-1,2-propanediol, hydrate)  
SGLT2
99.99%
Canagliflozin hemihydrate  
SGLT2
99.95%
Trilobatin
SGLT1
SGLT2
99.00%
SGLT2-IN-1  
SGLT2, IC50: 33 nM
99.82%
Tofogliflozin hydrate  
SGLT2
98.48%
Swertisin  
SGLT2
99.75%
Velagliflozin  
SGLT2
99.92%
Licogliflozin
SGLT1
SGLT2
98.03%
Dapagliflozin-d5  
SGLT2
98.01%
Ertugliflozin L-pyroglutamic acid  
SGLT2
99.84%
Remogliflozin etabonate
hSGLT1, Ki: 43.1 μM
rSGLT1, Ki: 8.57 μM
rSGLT2, Ki: 2.14 μM
hSGLT2, Ki: 1.95 μM
99.81%
Enavogliflozin  
SGLT2
98.43%
Canagliflozin-d4  
SGLT2
99.04%
Dapagliflozin impurity  
SGLT2
99.63%
Tianagliflozin  
SGLT2
99.96%
Luseogliflozin
SGLT1, IC50: 3990 nM
SGLT2, IC50: 2.26 nM
99.33%
Empagliflozin (Standard)  
SGLT2
Remogliflozin  
SGLT2
HSK0935  
SGLT2
Sergliflozin etabonate  
SGLT2
99.64%
Dapagliflozin-13C6-1  
SGLT2
Henagliflozin  
SGLT2
Luseogliflozin hydrate  
SGLT2
99.20%
SGLT1/2-IN-1
SGLT1, IC50: 15.72 mM
SGLT2, IC50: 3.67 mM
Pragliflozin-13C6  
SGLT2
YM543 free base  
SGLT2
Velagliflozin proline hydrate  
SGLT2
99.43%
Phloretin (Standard)
SGLT1
SGLT2
Atigliflozin
hSGLT1, IC50: 8.2 μM
hSGLT2, IC50: 10 nM
TA-1887
SGLT1, IC50: 230 nM
SGLT2, IC50: 1.4 nM
Kushenol K
SGLT1
SGLT2
Dapagliflozin ((2S)-1,2-propanediol, hydrate) (Standard)  
SGLT2
T-1095
hSGLT1, IC50: 22.8 μM
hSGLT2, IC50: 2.3 μM
YM-543  
SGLT2
Velagliflozin proline  
SGLT2
99.43%
fluoro-Dapagliflozin
hSGLT1, Ki: 330 nM
hSGLT2, Ki: 5.3 nM
Ertugliflozin (Standard)  
SGLT2
TP0438836
hSGLT1, IC50: 28 nM
hSGLT2, IC50: 7 nM
Ipragliflozin (Standard)  
SGLT2
Dapagliflozin (Standard)  
SGLT2
Canagliflozin (Standard)  
SGLT2
Sergliflozin-A
SGLT1
SGLT2
Olorigliflozin  
SGLT2
Phlorizin (Standard)
SGLT1
SGLT2
Dapagliflozin-d4  
SGLT2
Trilobatin (Standard)
SGLT1
SGLT2
galacto-Dapagliflozin
hSGLT1, Ki: 25000 nM
hSGLT2, Ki: 25 nM