2. GPCR/G Protein
  3. G Protein-coupled Receptor Kinase (GRK)
  4. GRK2 Inhibitor 2

GRK2 Inhibitor 2 (Compound 8h) 是一种 GRK2 抑制剂 (IC50: 19 nM)。GRK2 Inhibitor 2 还抑制 Aurora-A (IC50: 137 nM)。GRK2 Inhibitor 2 促进 GRK2 过表达 HEK293 细胞中 β-AR 介导的 cAMP 积累。GRK2 Inhibitor 2 可用于充血性心力衰竭 (HF) 的研究。

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GRK2 Inhibitor 2 Chemical Structure

GRK2 Inhibitor 2 Chemical Structure

CAS No. : 2592436-21-8

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GRK2 Inhibitor 2 相关抗体

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  • 生物活性

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生物活性

GRK2 Inhibitor 2 (Compound 8h) is a GRK2 inhibitor (IC50: 19 nM). GRK2 Inhibitor 2 also inhibits Aurora-A (IC50: 137 nM). GRK2 Inhibitor 2 promotes β-AR-mediated cAMP accumulation in GRK2-overexpressed HEK293 cells. GRK2 Inhibitor 2 can be used for research of congestive heart failure (HF)[1].

分子量

332.36

Formula

C19H16N4O2
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

GRK2 Inhibitor 2 相关分类

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  • Do most proteins show cross-species activity?

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Keywords:

GRK2 Inhibitor 22592436-21-8G Protein-coupled Receptor Kinase (GRK)congestive heart failureHFβ-ARcAMPHEK293Inhibitorinhibitorinhibit

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产品名称：
GRK2 Inhibitor 2
目录号：
HY-156863
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