2. Membrane Transporter/Ion Channel Neuronal Signaling
  3. iGluR Potassium Channel
  4. NR2B-selective NMDA receptor antagonist 1

NR2B-selective NMDA receptor antagonist 1 

目录号: HY-126123
产品使用指南

摩尔计算器

NR2B-selective NMDA receptor antagonist 1 (compound 29) 是 NR1/NR2B 受体的有效拮抗剂，对 NR1/NR2B NMDA 受体, hERG, α1-AdR 的 IC50 分别为 0.05 μM、0.73 μM、2.4 μM。NR2B-selective NMDA receptor antagonist 1 表现出有效的血脑屏障渗透性。

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NR2B-selective NMDA receptor antagonist 1 Chemical Structure

NR2B-selective NMDA receptor antagonist 1 Chemical Structure

CAS No. : 457897-92-6

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NR2B-selective NMDA receptor antagonist 1 相关抗体

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  • 生物活性

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生物活性

NR2B-selective NMDA receptor antagonist 1 (compound 29) is a potent antagonist of NR1/NR2B receptors, with IC50s of 0.05 μM, 0.73 μM, 2.4 μM to NR1/NR2B NMDA receptor, hERG, α1-AdR, respectivity. NR2B-selective NMDA receptor antagonist 1 exhibites efficient permeability across the blood–brain barrier[1].

体外研究
(In Vitro)

NR2B-selective NMDA receptor antagonist 1 (compound 29) (1 μM) 可以减弱 NMDA 诱导的 LDH 水平[1] 。

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

NR2B-selective NMDA receptor antagonist 1 相关抗体:
体内研究
(In Vivo)

NR2B-selective NMDA receptor antagonist 1 (compound 29) (30 mg/kg, i.p. once) 显示梗塞体积减少[1]。

MCE has not independently confirmed the accuracy of these methods. They are for reference only.
分子量

433.35

Formula

C18H22Cl2N2O4S
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

NR2B-selective NMDA receptor antagonist 1 相关分类

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This equation is commonly abbreviated as: C1V1 = C2V2

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

NR2B-selective NMDA receptor antagonist 1457897-92-6iGluRPotassium ChannelIonotropic glutamate receptorsKcsAblood–brain barrierNR2BInhibitorinhibitorinhibit

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