1. Signaling Pathways
  2. Cell Cycle/DNA Damage
    Stem Cell/Wnt
  3. Casein Kinase
  4. Casein Kinase Inhibitors

Casein Kinase Inhibitors

CK1

CK2

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

Casein Kinase Inhibitors & Chemicals
Product Name CK1 CK2 Purity
Silmitasertib  
CK2α, IC50: 1 nM
CK2α', IC50: 1 nM
99.94%
IWP-2
CK1δ, IC50: 40 nM
  99.51%
Emodin  
CK2α Wild-type, IC50: 5.9 μM (at ATP concentration is 50 μM)
CK2α Wild-type, IC50: 1.4 μM (at ATP concentration is 10 μM)
99.20%
Ellagic acid  
CK2, IC50: 40 nM
99.23%
TID43  
CK2, IC50: 0.3 μM
D4476
CK1, IC50: 0.3 μM
  99.94%
PF-670462 dihydrochloride
CKIδ, IC50: 14 nM
  99.96%
Silmitasertib sodium salt  
CK2α, IC50: 1 nM
CK2α', IC50: 1 nM
99.91%
TBB  
CK2, IC50: 0.15 μM (Human CK2)
99.31%
TMX-4116
CK1α
  99.50%
Casein Kinase inhibitor A51
CKIα
  98.58%
DMAT  
CK2, IC50: 0.13 μM (Human CK2)
98.09%
PF-4800567
CKIδ, IC50: 711 nM
  98.04%
SR-3029
CKIδ, IC50: 44 nM
  99.41%
FPFT-2216
CK1α
  99.35%
IC261
CKIδ, IC50: 1 μM
CkIα1, IC50: 16 μM
  99.54%
TAK-715
CK1δ
CK1ε
  99.73%
SGC-CK2-1  
CK2α, IC50: 36 nM
CK2α', IC50: 16 nM
99.41%
CKI-7 free base
CK1, IC50: 6 μM
CK1, Ki: 8.5 μM
  99.34%
TTP 22  
CK2, IC50: 100 nM
98.03%
BioE-1115  
CK2α, IC50: 10 μM
99.56%
CK1-IN-1
CKIδ, IC50: 15 nM
  99.35%
AMG-548 dihydrochloride
CK1
  99.91%
TA-01
CKIδ, IC50: 6.8 nM
  99.77%
PF-5006739
CK1δ, IC50: 3.9 nM
  99.56%
CK2/ERK8-IN-1  
CK2, IC50: 0.5 μM
CK2, Ki: 0.25 μM
≥99.0%
Hematein  
CKII, IC50: 0.74 μM
NCC007
CKIδ, IC50: 3.6 μM
CKIα, IC50: 1.8 μM
  99.73%
MRT00033659
CKIδ, IC50: 0.9 μM
  99.77%
Casein Kinase inhibitor A86
CKIα
  98.47%
Longdaysin
CKIδ, IC50: 8.8 μM
CKIα, IC50: 5.6 μM
  99.87%
TMX-4113
CK1α
  98.66%
LH846
CKIδ, IC50: 290 nM
CKIα, IC50: 2.5 μM
  98.04%
MU1742
CKIδ
  99.74%
CK2 inhibitor 2  
CK2, IC50: 0.66 nM
98.51%
Casein Kinase 2 Substrate Peptide  
CK2
98.47%
PI-828  
CK2α2, IC50: 1.127 μM
CK2, IC50: 149 nM
99.09%
SRPIN803  
CK2, IC50: 203 nM
99.17%
TBCA  
CK2, IC50: 110 nM
CK2, Ki: 77 nM
99.60%
A-3 hydrochloride
CK1, Ki: 80 μM
CK2, Ki: 5.1 μM
99.75%
BRD4/CK2-IN-1  
CK2, IC50: 230 nM
98.62%
AMG-548
CK1
  ≥99.0%
Casein kinase 1δ-IN-1
CKIδ
  99.91%
LY294002 hydrochloride  
CK2α2, IC50: 3.869 μM
CK2, IC50: 0.098 μM
CK2-IN-3  
CK2α, IC50: 1.51 μM
CK2α', IC50: 7.64 μM
Quinalizarin  
CK2, IC50: 110 nM
CK2, Ki: ~50 nM
Casein kinase 1δ-IN-3
CKIδ, pIC50: 6.5376 M
  99.93%
IQA  
CK2
Casein kinase 1δ-IN-4
CK1δ
  ≥98.0%
Casein kinase 1δ-IN-15
CK1δ, IC50: 0.045 μM
 
CK1-IN-2
CKIα, IC50: 123 nM
  99.54%
SR-4133
CK1δ, IC50: 10 μM
CK1ε, IC50: 58 nM
 
CK2/PIM1-IN-1  
CK2, IC50: 3.787 μM
CK1-IN-3
CK1δ, IC50: 2.22 μM
  99.00%
ON 108600  
CK2α2, IC50: 0.005 μM
CK2α1, IC50: 0.05 μM
99.73%
CK2 inhibitor 3  
CK2, IC50: 280 nM
Ellagic acid (hydrate)  
CK2, IC50: 40 nM
CK2, Ki: 20 nM
Casein kinase 1δ-IN-10
CK1δ
 
Casein kinase 1δ-IN-9
CK1δ
  ≥98.0%
Emodin (Standard)  
CK2α Wild-type
Multi-kinase-IN-6  
CK2, IC50: 0.09 μM
TMCB  
CK2α, Ki: 83 nM
CK2α', Ki: 21 nM
CKI-7
CK1, IC50: 6 μM
CK1, Ki: 8.5 μM
 
Casein Kinase II Receptor Peptide  
CK2, Km: 500 μM
SR-1277
CKIδ, IC50: 49 nM
 
AMG-548 hydrochloride
CK1
 
EGFR-IN-57  
CK2α, IC50: 0.171 μM
4,5,6,7-Tetrabromo-1H-benzimidazole  
CK2
Casein kinase 1δ-IN-5
CK1δ, IC50: 47 nM
 
(R)-DRF053 dihydrochloride
CK1, IC50: 14 nM