2. GPCR/G Protein Neuronal Signaling
  3. 5-HT Receptor
  4. CGS-12066 maleate

CGS-12066 maleate  (Synonyms: CGS-12066A马来酸盐)

目录号: HY-123704
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摩尔计算器

CGS-12066 (maleate) 是一种 5-HT 受体激动剂。 CGS-12066对5-HT1A、5-HT1B、5-HT1C 和 5-HT1D 具有激动作用， pEC50 值分别为 6.41、7.56、4.05 和 7.11。CGS-12066 可用于神经系统疾病的研究。

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CGS-12066 maleate Chemical Structure

CGS-12066 maleate Chemical Structure

CAS No. : 1350965-83-1

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CGS-12066 maleate 相关抗体

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查看 5-HT Receptor 亚型特异性产品:

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5-HT1 Receptor 5-HT2 Receptor 5-HT3 Receptor 5-HT4 Receptor 5-HT5 Receptor 5-HT6 Receptor 5-HT7 Receptor 5-HT Receptor

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

CGS-12066 (maleate) is a 5-HT receptor agonist. CGS-12066 has agonist effect for 5-HT1A , 5-HT1B ,5-HT1C and 5-HT1D with pEC50 values of 6.41, 7.56, 4.05 and 7.11, respectively. CGS-12066 can be used for the research of neurological disease[1].
IC50 & Target

pEC50: 6.41 (5-HT1A), 7.56 (5-HT1B), 4.05 (5-HT1C) and 7.11 (5-HT1D)[1].
pKD: 7.19 (5-HT1A), 6.94 (5-HT1B), 4.89 (5-HT1C) and 7.49 (5-HT1D)[1].
体外研究
(In Vitro)

CGS-12066 (maleate) 对 5-HT1A、5-HT1B、5-HT1C 和 5-HT1D 具有激动作用，pEC50 值分别为 6.41、7.56、4.05 和 7.11[1]。
CGS-12066 (maleate) 对 5-HT1A、5-HT1B、5-HT1C和5-HT1D具有激动作用，pKD 值分别为 7.19、6.94、4.89 和 7.49[1]。
CGS-12066 (maleate) 以低效能刺激肌醇磷酸盐的积累[1]。
CGS-12066 (maleate) 作为部分激动剂抑制小腿黑质毛喉素刺激的腺苷酸环化酶活性[1]。

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

CGS-12066 maleate 相关抗体:
分子量

450.41

Formula

C21H21F3N4O4
CAS 号
中文名称

CGS-12066A马来酸盐
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

CGS-12066 maleate 相关分类

  • 摩尔计算器

  • 稀释计算器

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

CGS-120661350965-83-1CGS-12066A马来酸盐CGS12066CGS 120665-HT ReceptorSerotonin Receptor5-hydroxytryptamine Receptor5-HT receptorneurological disease5-HT1A5-HT1B5-HT1C5-HT1DInhibitorinhibitorinhibit

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