2. GPCR/G Protein
  3. Adenosine Receptor
  4. A1/A3 AR antagonist 1

A1/A3 AR antagonist 1 (compound 10) 是一种有效的腺苷酸 1 (A1) 和腺苷酸 3 (A3) 受体双重拮抗剂，对人 A1、人 A3 和大鼠 A1 的 Ki 分别为 36.7 nM、25.4 nM 和 1.47 nM。A1/A3 AR antagonist 1 可用于肾衰竭、炎症性肺部疾病和阿尔茨海默症的研究。

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A1/A3 AR antagonist 1 Chemical Structure

A1/A3 AR antagonist 1 Chemical Structure

CAS No. : 312929-49-0

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A1/A3 AR antagonist 1 相关抗体

Top Publications Citing Use of Products

查看 Adenosine Receptor 亚型特异性产品:

查看所有亚型
Adenosine A1 receptor (A1R) Adenosine A2A receptor (A2AR) Adenosine A2B receptor (A2BR) Adenosine A3 receptor (A3R)

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

A1/A3 AR antagonist 1 (compound 10) is a potent adenosine 1 (A1) and adenosine 3 (A3) receptor dual antagonist with Kis of 36.7 nM, 25.4 nM and 1.47 nM for human A1, human A3 and rat A1, respectively. A1/A3 AR antagonist 1 can be used for researching kidney failure, inflammatory pulmonary diseases, and Alzheimer’s disease[1].

IC50 & Target[1]

human A1

36.7 nM (Ki)

rat A1

1.47 nM (Ki)

human A3

25.4 nM (Ki)

分子量

414.48

Formula

C24H18N2O3S
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

A1/A3 AR antagonist 1 相关分类

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

A1/A3 AR antagonist 1312929-49-0Adenosine ReceptorP1 receptorKidney failureInflammatory pulmonary diseasesAlzheimer’s diseaseInhibitorinhibitorinhibit

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