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Metabolism/Protease Compound Library

Cat. No.: HY-L012
Library Contents: XLSX PDF

A unique collection of 795 Metabolism/Protease-related small molecules for high throughput screening (HTS) and high content screening (HCS).

Metabolism/Protease Compound Library
Size (Pre-dissolved DMSO or Solid) Price Stock
30 μL/well (10 mM solution) Get quote In-stock
50 μL/well (10 mM solution) Get quote In-stock
100 μL/well (10 mM solution) Get quote In-stock
250 μL/well (10 mM solution) Get quote In-stock

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  • Description

  • Product Details

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  • Contents

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Description
& Advantages

•   A unique collection of 795 Metabolism/Protease-related small molecules for high throughput screening (HTS) and high content screening (HCS).

•   Targets such as PDE, Cytochrome P450, HMG-CoA Reductase, DPP4, Proteasome, HCV Protease, IDO, Cathepsin, MMP, etc.

•   A useful tool for drug discovery of metabolism-related diseases.

•   Bioactivity and safety confirmed by preclinical research and clinical trials. Some inhibitors have been approved by FDA.

•   Structurally diverse, medicinally active, and cell permeable.

•   More detailed compound information with structure, IC50, and brief introduction.

•   NMR and HPLC validated to ensure high purity and quality.

•   All compounds are in stock and continuously updated.

Product Details
Formulation:
A collection of 795 Metabolism/Protease related compounds supplied as pre-dissolved DMSO solutions or Solid
Container:
96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode
Storage:
-80°C
Shipping:
Blue ice
Composition

Metabolism/Protease Compound Library

Source: MedChem Express

Contents of Metabolism/Protease Compound Library

Plate layout: HY-L012-1

1 2 3 4 5 6 7 8 9 10 11 12
a Empty BAY-1436032 NSC 663284 KNK437 AM-2394 SZL P1-41 WWL70 CL-82198 A 922500 FCCP Odanacatib Empty
b Empty TM5275 (sodium) TPI-1 Benzophenonetetracarboxylic acid PD150606 CD437 Flopropione Ribitol (-)-(S)-Equol (±)-Equol Stibogluconate (sodium) Empty
c Empty Urolithin A BVT948 BVT948 SYP-5 ML348 ML349 RA190 Norverapamil (hydrochloride) IDO-IN-2 2-PMPA Empty
d Empty CHS-828 SR12813 Hypotaurine Kynurenic acid Quinolinic acid (R)-Serine KRIBB11 GCN2-IN-1 CDD3505 MK-8617 Empty
e Empty Sarcosine NQ301 TOFA AR7 Allopregnanolone UK-371804 XMD16-5 Vadadustat DMU2139 Cilostamide Empty
f Empty Deoxycytidine triphosphate Cyclo(his-pro) N-(5-Aminopentyl)acetamide DL-Homocysteine thiolactone (hydrochloride) Nicotinamide N-oxide Docosatrienoic Acid O-Acetylserine SDMA 4-Acetamidobutanoic acid 2-(Methylamino)-1H-purin-6(7H)-one Empty
g Empty Iberin L-DABA Vanilpyruvic acid SR9238 SR0987 SR-18292 HTS01037 BMS-986205 TRC051384 TM5441 Empty
h Empty UAMC00039 (dihydrochloride) GLPG1690 DKM 2-93 BMS-309403 Prostaglandin E2 6-Biopterin Tanespimycin BIIB021 Luminespib Bortezomib Empty

Plate layout: HY-L012-2

1 2 3 4 5 6 7 8 9 10 11 12
a Empty PX-478 Telaprevir Boceprevir Danoprevir Mericitabine Simeprevir Edoxaban (tosylate monohydrate) Betrixaban Dabigatran etexilate Dabigatran etexilate (mesylate) Empty
b Empty Linagliptin Saxagliptin Tarenflurbil ML-030 ABT-702 dihydrochloride 1-Aminobenzotriazole Stiripentol Methylmalonate Raltegravir Raltegravir (potassium salt) Empty
c Empty PKM2-IN-1 3-Methoxytyramine hydrochloride 3-Methoxytyramine CTS-1027 L-Kynurenine BAY 73-6691 racemate Ixazomib citrate Ixazomib Delanzomib Carfilzomib Empty
d Empty Daclatasvir (dihydrochloride) Daclatasvir GSK256066 AM580 Cobicistat Tipifarnib Orteronel Darapladib Ro 28-1675 T0901317 Empty
e Empty GW3965 (hydrochloride) LXR-623 4-Butylresorcinol Tetrahydrobiopterin UVI 3003 LY2955303 Cilomilast DPP-IV-IN-2 URB-597 LY2183240 Empty
f Empty GSK2033 Apararenone Cilofexor Fexaramine Pifithrin-μ VER-155008 VER-82576 BRL-50481 Arachidonic acid D4-abiraterone Empty
g Empty Crisaborole Pyributicarb 1-Linoleoyl Glycerol PF-05180999 1-Ethynylnaphthalene GSTO1-IN-1 Mitochonic acid 5 Retagliptin Phosphate TFAP BN82002 Empty
h Empty Urocanic acid Maltotriose p-Hydroxymandelic acid N-Acetylornithine 1-Methyladenosine 25-Hydroxycholesterol 5-Methylcytidine Galactose 1-phosphate Potassium salt Asymmetric dimethylarginine p-Synephrine Empty

Plate layout: HY-L012-3

1 2 3 4 5 6 7 8 9 10 11 12
a Empty trans-trans-Muconic acid 3-Methyladipic acid Leucyl-phenylalanine Ureidopropionic acid 4-Guanidinobutanoic acid Citraconic acid Aminoadipic acid Nicotinuric acid Anserine Petroselinic acid Empty
b Empty N-Methylhydantoin DL-Dopa 3-Hydroxyisovaleric acid 3-Methylglutaric acid Nepsilon-Acetyl-L-lysine N-Acetyl-L-aspartic acid Alvespimycin (hydrochloride) Apremilast Torcetrapib Anacetrapib Empty
c Empty Oprozomib Aliskiren Aliskiren (hemifumarate) INT-747 T-5224 PI-1840 TCS 401 IBMX SB-3CT C75 Empty
d Empty C75 (trans) Angiotensin (1-7) Balipodect Oltipraz Velpatasvir RVT-501 ML228 FIPI STF-118804 AEBSF Empty
e Empty JNJ-42041935 PF-05175157 PF-04620110 LX1606 (Hippurate) LX1606 Celastrol ONX-0914 Avasimibe Talabostat (mesylate) Dolutegravir Empty
f Empty Dolutegravir (sodium) BMS-707035 Nepicastat (hydrochloride) Vinpocetine PYR-41 PYZD-4409 Oseltamivir (acid) Evacetrapib PF-8380 Varespladib Empty
g Empty SR1001 FG-4592 KW-2478 Debio 0932 U-104 Clinofibrate Cladribine Dutasteride Ezatiostat Finasteride Empty
h Empty LW6 Quinacrine (dihydrochloride) Sitagliptin Sitagliptin (phosphate monohydrate) Ursodiol 2-Deoxy-D-glucose IDO-IN-7 Ombitasvir Zileuton Bexarotene Empty

Plate layout: HY-L012-4

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Milrinone Olprinone (Hydrochloride) Febuxostat Isavuconazole Entacapone Vildagliptin PF-04457845 PF-3845 SR3335 SR1078 Empty
b Empty AT13387 Lopinavir Biochanin A (S)-Glutamic acid Retinoic acid DHEA Tamibarotene Fluvastatin (sodium) Choline Fenofibrate Elvitegravir Empty
c Empty TRO 19622 Palifosfamide Teneligliptin Teneligliptin (hydrobromide) Topiroxostat Anagliptin Gemigliptin Dalcetrapib N6022 Bay 60-7550 Empty
d Empty Sildenafil Sildenafil (citrate) Apoptozole Balicatib Isotretinoin O-Phospho-L-serine Lonafarnib Oglemilast NVP-HSP990 GSK 650394 Empty
e Empty EMD638683 Ganetespib Geldanamycin JZL 184 JZL195 Tiplaxtinin CP-640186 (hydrochloride) E-64 Nelfinavir (Mesylate) Fenretinide Empty
f Empty Tazarotene AHU-377 AHU-377 (hemicalcium salt) Trelagliptin Trelagliptin (succinate) 5-Iodotubercidin PF-04447943 Roflumilast IOX2 Zardaverine Empty
g Empty Salubrinal Cabotegravir Ledipasvir Ledipasvir (acetone) Ledipasvir (D-tartrate) FG-2216 Alvelestat Bivalirudin (Trifluoroacetate) TTNPB IDO5L Empty
h Empty INCB 024360 PluriSln 1 AGI-6780 GM6001 NSC 405020 GSK 2830371 BAY 87-2243 SF1670 Atglistatin FTI-277 (hydrochloride) Empty

Plate layout: HY-L012-5

1 2 3 4 5 6 7 8 9 10 11 12
a Empty DMOG Sal003 AZD7545 BMS-303141 L-778123 (hydrochloride) Tolrestat Skp2 Inhibitor C1 Dafadine-A Rolipram (R)-(-)-Rolipram Empty
b Empty 5'-Methylthioadenosine SW033291 SR9243 Saquinavir (Mesylate) Saquinavir Darunavir Darunavir (Ethanolate) Fenofibrate Clozapine (N-oxide) Atazanavir (sulfate) Empty
c Empty Dabigatran (ethyl ester) Atorvastatin (hemicalcium salt) Racecadotril Tolcapone Mevastatin Amprenavir Sivelestat Sivelestat (sodium tetrahydrate) Cortisone Cilostazol Empty
d Empty Simvastatin Rosuvastatin (Calcium) Clarithromycin ZLN005 sn-Glycero-3-phosphocholine 2'-Deoxyguanosine Daprodustat AGI-5198 LCZ696 Omapatrilat Empty
e Empty Leupeptin (hemisulfate) Avanafil Udenafil L-Thyroxine 3-Indoleacetic acid TZ9 TEPP-46 PU-WS13 CPDA Enasidenib Empty
f Empty Enasidenib (mesylate) Endoxifen (hydrochloride) Lipoic acid VR23 Ivosidenib (R,S)-Ivosidenib NCT-501 KC7F2 Alda-1 Aldose reductase-IN-1 Empty
g Empty KML29 Adjudin 3-Methyladenine HA130 DASA-58 TMS GSK864 BEC (hydrochloride) JNJ-42165279 (-)-p-Bromotetramisole (oxalate) Empty
h Empty PD 151746 Indirubin-3'-monoxime PRT4165 BMS-779788 3-Bromopyruvic acid AM 3112 Methoxsalen (S)-Leucic acid (S)-2-Hydroxy-3-phenylpropanoic acid Clemizole (hydrochloride) Empty

Plate layout: HY-L012-6

1 2 3 4 5 6 7 8 9 10 11 12
a Empty T863 Ethylmalonic acid L-Hydroxyproline Octanoic acid 5-Amino-3H-imidazole-4-Carboxamide D-Alanine (-)-Aspartic acid GW 4064 Apixaban DGAT-1 inhibitor 2 Empty
b Empty A939572 3-Methylxanthine FK866 Rivaroxaban WAY-362450 2-Amino-1-phenylethanol Epalrestat Carboxypeptidase G2 (CPG2) Inhibitor CPA inhibitor TOK-001 Empty
c Empty Abiraterone Otamixaban GSK256066 (2,2,2-trifluoroacetic acid) D609 SPK-601 Abiraterone (acetate) VX-222 L-Pyroglutamic acid Vitamin D2 Chenodeoxycholic Acid Empty
d Empty 5-R-Rivaroxaban Dabigatran (ethyl ester hydrochloride) FAAH-IN-2 Ritonavir Nortadalafil Tadalafil Pentostatin Alogliptin (Benzoate) Cilazapril (monohydrate) Malotilate Empty
e Empty N-Acetyl-D-glucosamine Adenosine monophosphate Doxofylline Melatonin Adapalene Benazepril (hydrochloride) Edaravone Ketoconazole (+)-Ketoconazole Acitretin Empty
f Empty Dorzolamide (hydrochloride) Diphylline Perindopril (erbumine) Bestatin Aminophylline Estradiol Alpha-Estradiol Niacin Pitavastatin (Calcium) Nicotinamide Empty
g Empty Pregnenolone Adenine Cytidine Pravastatin (sodium) Lithocholic acid Nafamostat (mesylate) Pimobendan Metolazone Acetylcysteine Ethynyl Estradiol Empty
h Empty Orlistat Allopurinol Adenosine Enalaprilat (dihydrate) Estrone Disulfiram Eplerenone Gemfibrozil Thiabendazole Ramipril Empty

Plate layout: HY-L012-7

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Dipyridamole Irsogladine Enalapril (maleate) Menadione Taurine Memantine (hydrochloride) Captopril Argatroban (monohydrate) Moexipril (hydrochloride) Fosinopril (sodium) Empty
b Empty Temocapril (hydrochloride) Gabexate (mesylate) Dextrose (S)-(+)-Rolipram Dichlorphenamide D-Sorbitol Estriol Ozagrel Ozagrel (sodium) Vardenafil (hydrochloride) Empty
c Empty NAD+ Dopamine (hydrochloride) Hydralazine (hydrochloride) Quinapril (hydrochloride) Tioxolone Lonidamine PMSF Creatinine Anagrelide (hydrochloride) Methazolamide Empty
d Empty Brinzolamide Trandolapril Fondaparinux (sodium) Levobupivacaine (hydrochloride) Zofenopril (calcium) Eicosapentaenoic Acid Indinavir (sulfate) Azelaic acid Pentoxifylline Ibudilast Empty
e Empty Teprenone Acetazolamide Theophylline Tebuconazole Hexylresorcinol L-SelenoMethionine 4-Aminobenzoic acid Tilorone (dihydrochloride) N-Acetylprocainamide Benzbromarone Empty
f Empty Cotinine Tetramisole (hydrochloride) Alrestatin Fludrocortisone (acetate) Histamine Carprofen Metyrapone Protoporphyrin IX 4-Aminohippuric acid Proadifen (hydrochloride) Empty
g Empty Retinol 4-Aminoantipyrine Salicylanilide i-Inositol Ethoxyquin Canrenone Uridin Imidapril (hydrochloride) Deoxyarbutin Chlorzoxazone Empty
h Empty Deoxycorticosterone (acetate) Serotonin hydrochloride Ethoxzolamide cAMP Corticosterone Pyridoxal phosphate Rotenone Spermidine Carbosulfan Lactose Empty

Plate layout: HY-L012-8

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Uric acid Tryptamine 2-Aminobenzenesulfonamide Docosahexaenoic Acid ATP Stearic acid 2'-Deoxycytidine 2'-Deoxyuridine Glutathione oxidized Tartaric acid (disodium dihydrate) Empty
b Empty Sodium orthovanadate Glycylglycine β-Nicotinamide mononucleotide Iloperidone metabolite Hydroxy Iloperidone Omeprazole metabolite Omeprazole sulfide Norgestimate metabolite Norelgestromin N-Desmethylclozapine Epiandrosterone N-Acetylneuraminic acid 6-Aminopyrimidin-2(1H)-one Empty
c Empty PCL 016 Regorafénib N-oxyde (M2) Uracil L-Alloisoleucine Icariin Daidzin Arctigenin Ginsenoside Rd Chlorogenic acid Ginkgolic Acid Empty
d Empty Dimethylfraxetin Hypoxanthine Inosine Guanosine Vanillin Isoliquiritigenin Coenzyme Q10 Diosmetin Stigmasterol Tanshinone I Empty
e Empty Taxifolin Theobromine Naringin Oleanolic Acid Orotic acid Magnolol Caffeic acid 18β-Glycyrrhetinic acid Arbutin Baicalein Empty
f Empty Nordihydroguaiaretic acid D-Galactose (-)-Epigallocatechin L-Alanine β-Alanine Cordycepin Paeoniflorin Stachydrine Salvianolic acid A Bilirubin Empty
g Empty Cholic acid L-Methionin Bergapten D-Mannitol D-Mannose Galangin Homovanillic acid L-Glutamine L-Citrulline L-Cystine Empty
h Empty β-Carotene Succinic acid Astragaloside IV Progesterone L-Arginine α-Lipoic Acid Gentiopicroside Lovastatin Morroniside Xylose Empty

Plate layout: HY-L012-9

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Allantoin Oroxylin A Doxycycline (hyclate) Umbelliferone Hydrocortisone Deoxycholic acid Ginsenoside F1 Cinnamic acid Mulberroside A Dicoumarol Empty
b Empty L-Serine L-Aspartic acid L-Asparagine Schisandrin A Glucosamine (hydrochloride) Coptisine (chloride) Ginkgolide C Phytic acid Shikonin Palmitic acid Empty
c Empty L-Hisidine (20S)-Protopanaxatriol AKBA Tetrahydrocurcumin Ginsenoside C-K Androsterone Xanthohumol Thymidine Apigenin 2-Methoxybenzoic acid Empty
d Empty Glycocholic acid Glycoursodeoxycholic acid Citric acid Oxyresveratrol (-)-Fucose Loureirin B Pyrogallol 4',5-Dihydroxyflavone Propylparaben Taurochenodeoxycholic acid Empty
e Empty Glycochenodeoxycholic acid 11beta-Hydroxyprogesterone Cholesteryl behenate Palmitelaidic Acid p-Hydroxycinnamic acid D-Arabitol [Leu5]-Enkephalin 3,4-Dihydroxybenzeneacetic acid 2,5-Dihydroxybenzoic acid Pyrrole-2-carboxylic acid Empty
f Empty 2,5-Furandicarboxylic acid L-Homoserine 4-Hydroxy-3-methylbenzoic acid 2-(4-Methoxyphenyl)acetic acid Pentadecanoic acid 5-Hydroxymethyluracil 5-Hydroxymethyl-2-furancarboxylic acid 3-Methyl-2-oxobutanoic acid Tyramine 3-Oxopentanedioic acid Empty
g Empty 2-Oxobutanoic acid H-Phe-Phe-OH 2-Hydroxy-3-methylbutanoic acid 5-Hydroxyindole-3-acetic acid H-HoArg-OH H-Tyr(3-I)-OH Glutaric acid DL-Homocystine 5-Methyluridine Terephthalic acid Empty
h Empty 4,6-Dioxoheptanoic acid 2-Methylsuccinic acid Creatine Thymine DL-Norvaline H-Abu-OH Adenosine 5'-diphosphate Xanthosine L-Homocystine Dodecanedioic acid Empty

Plate layout: HY-L012-10

1 2 3 4 5 6 7 8 9 10 11 12
a Empty N-Acetyl-L-tyrosine H-D-Trp-OH 2-Oxo-3-phenylpropanoic acid 2,4-Dihydroxybenzoic acid 3-Amino-4-methylpentanoic acid H-HoPro-OH 4-Methylcatechol 4-Ethylphenol 3-Amino-2-methylpropanoic acid 2-Ketoglutaric acid Empty
b Empty Undecanedioic acid Ac-Arg-OH Decanedioic acid 1,3-Dimethyluric acid 2-(2-Methylbenzamido)acetic acid 3-Indolepropionic acid Octanedioic acid 3-Hydroxymandelic Acid Desaminotyrosine N-Isovaleroylglycine Empty
c Empty 3,5-Dihydroxybenzoic acid 2-Hydroxyphenylacetic acid 2-Phenylpropionic acid L-(+)-Arabinose 2-Hydroxy-2-methylbutanoic acid Fumaric acid Glycolic acid Hippuric acid L-Gulono-1,4-lactone trans-Aconitic acid Empty
d Empty H-Gly-Pro-OH 1-Methyl-L-histidine 3-Methyl-L-histidine L-Ornithine Hydrochloride 7-Methylxanthine Xanthine Adipic acid 2-Methylpentanedioic acid L-Homocitrulline DL-Glyceric Acid Empty
e Empty Hexadecanedioic acid 2-Guanidinoacetic acid L-Arabinitol 2'-Deoxyadenosine 3-Chloro-L-tyrosine Phenylacetylglutamine (S)-3-Hydroxybutanoic acid (R)-3-Hydroxybutanoic acid (±) Anabasine L-Norleucine Empty
f Empty 3-Hydroxypicolinic acid N-Acetylglycine 2-Naphthol NSC 16590 D(-)-2-Aminobutyric acid Pyrocatechuic acid L-Proline 4-Hydroxybenzoic acid p-Hydroxybenzaldehyde L-Cysteine Empty
g Empty Maleic Acid Dulcite L-Lactic acid N-Methylsarcosine Pipecolic acid 3-Methoxybenzoic acid 3,4-Dimethoxyphenylacetic acid Pyruvic acid 2,6-Dihydroxybenzoic acid Levulinic acid Empty
h Empty Glycine (S)-2-Hydroxysuccinic acid Hydrocinnamic acid Pimelic acid Malic acid Empty Empty Empty Empty Empty Empty
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产品名称:
Metabolism/Protease Compound Library
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HY-L012
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