1. GPCR/G Protein
    Neuronal Signaling
  2. Opioid Receptor

LY-2940094 

目录号: HY-114452 纯度: 99.56%
产品使用指南

LY2940094是有效,选择性,有口服活性的 孤菲肽受体 (NOP) 拮抗剂,Ki为0.105 nM。

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LY-2940094 Chemical Structure

LY-2940094 Chemical Structure

CAS No. : 1307245-86-8

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Size Price Stock Quantity
10 mM * 1 mL in DMSO ¥4950 In-stock
5 mg ¥4500 In-stock
10 mg ¥7500 In-stock
25 mg ¥15000 In-stock
50 mg ¥21000 In-stock
100 mg ¥33000 In-stock
200 mg   Get quote  
500 mg   Get quote  

* Please select Quantity before adding items.

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Description

LY2940094 is a potent, selective and orally available nociceptin receptor (NOP) antagonist with an Ki of 0.105 nM.

IC50 & Target

Ki: 0.105 nM (NOP)[1]

Solvent & Solubility
In Vitro: 

DMSO : 41.67 mg/mL (86.64 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.0792 mL 10.3959 mL 20.7917 mL
5 mM 0.4158 mL 2.0792 mL 4.1583 mL
10 mM 0.2079 mL 1.0396 mL 2.0792 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

    Solubility: ≥ 2.08 mg/mL (4.32 mM); Clear solution

  • 2.

    Add each solvent one by one:  10% DMSO    90% corn oil

    Solubility: ≥ 2.08 mg/mL (4.32 mM); Suspended solution

  • 3.

    Add each solvent one by one:  10% DMSO    90% (20% SBE-β-CD in saline)

    Solubility: ≥ 2.08 mg/mL (4.32 mM); Clear solution

References
Molecular Weight

480.96

Formula

C₂₂H₂₃ClF₂N₄O₂S

CAS No.

1307245-86-8

SMILES

OCC1=CC=CN=C1N2N=C(C)C(CN3CCC4(C5=C(C=C(Cl)S5)C(F)(F)CO4)CC3)=C2

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Shipping

Room temperature in continental US; may vary elsewhere

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The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Inquiry Information

产品名称:
LY-2940094
目录号:
HY-114452
需求量:

LY-2940094

Cat. No.: HY-114452