Product Name |
α adrenergic receptor |
β adrenergic receptor |
Purity |
Isoprenaline hydrochloride |
|
|
99.86% |
Norepinephrine |
α1-adrenergic receptor
α2-adrenergic receptor
|
Beta-1 adrenergic receptor
|
99.33% |
Zenidolol hydrochloride |
|
|
99.76% |
Phenylephrine |
|
|
99.52% |
Propranolol hydrochloride |
|
|
99.97% |
ORM-10921 free base |
Alpha-2C adrenergic receptor, Ki: 1.4 nM
|
|
|
CL 316243 |
|
|
99.67% |
D-Mannitol |
|
Beta-3 adrenergic receptor
|
99.93% |
Phenylephrine hydrochloride |
|
|
99.76% |
Norepinephrine hydrochloride |
α1-adrenergic receptor
α2-adrenergic receptor
|
Beta-1 adrenergic receptor
|
99.95% |
Propranolol |
|
|
99.87% |
Metoprolol |
|
|
99.94% |
Atenolol |
|
Beta-1 adrenergic receptor, Ki: 697 nM
|
99.94% |
Prazosin hydrochloride |
|
|
99.86% |
Clozapine |
α2-adrenergic receptor, Ki: 51 nM (Inhibitor)
|
|
99.97% |
Norepinephrine bitartrate monohydrate |
α1-adrenergic receptor
α2-adrenergic receptor
|
Beta-1 adrenergic receptor
|
99.75% |
Dexmedetomidine |
α2-adrenergic receptor, Ki: 1.08 nM
|
|
99.93% |
Nadolol |
|
|
99.97% |
Mirabegron |
|
|
99.90% |
Yohimbine |
|
|
99.91% |
Phenylacetylglycine |
|
|
99.63% |
Salmeterol |
|
β3 adrenoceptor, pEC50: 5.9
β2 adrenoceptor, pEC50: 9.6
β1 adrenoceptor, pEC50: 6.1
|
99.91% |
Dexmedetomidine hydrochloride |
α2-adrenergic receptor, IC50: 1.08 nM
|
|
99.93% |
Salbutamol |
|
|
99.92% |
SR59230A |
|
|
≥98.0% |
Dobutamine hydrochloride |
|
|
99.91% |
(S)-Timolol maleate |
|
|
99.89% |
Phentolamine mesylate |
|
|
99.87% |
Paliperidone |
|
|
99.69% |
Labetalol |
|
|
99.88% |
Vilanterol trifenatate |
|
|
99.61% |
SR59230A hydrochloride |
|
|
99.87% |
Octopamine hydrochloride |
|
|
99.65% |
Guanfacine hydrochloride |
|
|
99.96% |
Tamsulosin |
|
|
99.77% |
L748337 |
|
Beta-2 adrenergic receptor, Ki: 204 nM
Beta-1 adrenergic receptor, Ki: 390 nM
Beta-3 adrenergic receptor, Ki: 4 nM
|
99.67% |
Bisoprolol hemifumarate |
|
Beta-1 adrenergic receptor
|
99.73% |
Mirtazapine |
α2-adrenergic receptor, pKi: 6.95
|
|
99.94% |
Terbutaline sulfate |
|
|
99.95% |
Fenoterol hydrobromide |
|
|
99.90% |
Atipamezole hydrochloride |
|
|
99.97% |
Nefazodone hydrochloride |
|
|
99.87% |
Doxazosin mesylate |
|
|
98.34% |
Pronethalol |
|
|
99.73% |
Indacaterol |
|
|
99.98% |
Salbutamol hemisulfate |
|
|
≥98.0% |
Metoprolol succinate |
|
|
99.90% |
Reboxetine mesylate |
|
|
99.90% |
Methyldopa hydrate |
|
|
99.95% |
Indacaterol maleate |
|
|
99.81% |
BI-167107 |
|
|
99.98% |
Vibegron |
|
β3 adrenoceptor, EC50: 1.1 nM
|
98.82% |
Acebutolol hydrochloride |
|
|
99.97% |
Vilanterol |
|
|
99.30% |
Naftopidil |
Alpha-1A adrenergic receptor, Ki: 3.7 nM
Alpha-1D adrenergic receptor, Ki: 1.2 nM
Alpha-1B adrenergic receptor, Ki: 20 nM
|
|
98.47% |
Idazoxan hydrochloride |
|
|
99.32% |
Midodrine hydrochloride |
|
|
99.49% |
Brimonidine |
|
|
99.99% |
(R)-Propranolol hydrochloride |
|
|
99.36% |
JP1302 dihydrochloride |
human α2C-adrenoceptor, Ki: 28±2 nM
rodent α2D-adrenoceptor, Ki: 1700±200 nM
human α2A-adrenoceptor, Ki: 3150±50 nM
human α2B-adrenoceptor, Ki: 1470±130 nM
|
|
99.62% |
Medetomidine hydrochloride |
α1-adrenergic receptor, Ki: 1750 nM
α2-adrenergic receptor, Ki: 1.08 nM
|
|
99.92% |
Lubabegron |
|
|
98.21% |
Olodaterol |
|
β2 adrenoceptor, EC50: .1 nM
|
98.48% |
Asenapine |
α1-adrenergic receptor, pKi: 8.9
Alpha-2A adrenergic receptor, pKi: 8.9
Alpha-2C adrenergic receptor, pKi: 8.9
Alpha-2B adrenergic receptor, pKi: 9.5
|
|
99.93% |
Practolol |
|
|
99.78% |
Butaxamine hydrochloride |
|
Beta-2 adrenergic receptor
|
99.87% |
Bufuralol |
|
|
99.17% |
Salmeterol xinafoate |
|
β3 adrenoceptor, pEC50: 5.9
β2 adrenoceptor, pEC50: 9.6
β1 adrenoceptor, pEC50: 6.1
|
99.96% |
Olodaterol hydrochloride |
|
β2 adrenoceptor, EC50: .1 nM
|
98.87% |
Synephrine |
|
|
≥98.0% |
Blonanserin |
α1-adrenergic receptor, Ki: 26.7 (Rat nM
α2-adrenergic receptor, Ki: 530 (Rat c nM
|
|
99.62% |
Ecopipam hydrochloride |
Alpha-2A adrenergic receptor, Ki: 731 nM
|
|
99.46% |
Medetomidine |
α1-adrenergic receptor, Ki: 1750 nM
α2-adrenergic receptor, Ki: 1.08 nM
|
|
99.99% |
Levobunolol hydrochloride |
|
|
99.89% |
Isoferulic acid |
|
|
99.82% |
(S)-(-)-Propranolol hydrochloride |
|
|
≥98.0% |
Bevantolol hydrochloride |
|
|
98.98% |
Carazolol |
|
β3 adrenoceptor
β2 adrenoceptor
β1 adrenoceptor
|
99.71% |
Oxprenolol hydrochloride |
|
β-adrenoceptor, Ki: 7.1 nM
|
99.86% |
Terbutaline |
|
Beta-2 adrenergic receptor
|
99.65% |
Dapiprazole hydrochloride |
|
|
99.87% |
LY 344864 |
rat α1-adrenergic receptor, Ki: 5.06 μM
rat α2-adrenergic receptor, Ki: 3.69 μM
|
|
98.93% |
Harmane |
α2-adrenergic receptor, IC50: 18 μM
|
|
99.84% |
Phentolamine |
|
|
99.89% |
ARC 239 dihydrochloride |
Alpha-2B adrenergic receptor
|
|
99.57% |
Metipranolol |
|
β2 adrenoceptor, pA2: 8.4
β1 adrenoceptor, pA2: 8.3
|
98.36% |
Talipexole dihydrochloride |
α2-adrenergic receptor, IC50: 25 nM
|
|
99.80% |
Isoetharine mesylate |
|
|
99.87% |
Urapidil hydrochloride |
α1-adrenergic receptor, pIC50: 6.13
α2-adrenergic receptor, pIC50: 4.38
|
|
99.97% |
Ecopipam hydrobromide |
Alpha-2A adrenergic receptor, Ki: 731 nM
|
|
≥99.0% |
Synephrine hydrochloride |
|
|
99.66% |
Xylometazoline hydrochloride |
Alpha-1A adrenergic receptor, Ki: 0.05 μM
Alpha-2A adrenergic receptor, Ki: 0.88 μM
Alpha-2C adrenergic receptor, Ki: 0.19 μM
Alpha-2B adrenergic receptor, Ki: 1.7 μM
Alpha-1D adrenergic receptor, Ki: 0.15 μM
Alpha-1B adrenergic receptor, Ki: 0.30 μM
|
|
99.58% |
BMY-14802 hydrochloride |
|
|
98.02% |
(RS)-Butyryltimolol |
|
|
≥98.0% |
Ajmalicine |
α1-adrenergic receptor
α2-adrenergic receptor
|
|
99.39% |
Methyldopate |
|
|
98.01% |
Bufuralol hydrochloride |
|
|
≥99.0% |
Tasipimidine sulfate |
human α2C-adrenoceptor, pEC50: 6.29
rodent α2D-adrenoceptor, pEC50: 6.56
human α2A-adrenoceptor, pEC50: 7.57
human α2B-adrenoceptor, pEC50: 6.00
|
|
99.46% |
A-61603 |
|
|
≥98.0% |
Arformoterol |
|
Beta-2 adrenergic receptor, Kd: 2.9 nM
|
99.96% |
Dicentrine |
|
|
99.38% |
Tamsulosin hydrochloride |
|
|
99.81% |
Spiroxatrine |
|
|
99.18% |
Bupranolol |
|
|
99.44% |
ST1936 |
α1-adrenergic receptor, Ki: 390 nM (rat)
α2-adrenergic receptor, Ki: 300 nM (rat)
α2-adrenergic receptor, Ki: 300 nM (human)
|
|
99.70% |
Metaterol |
|
|
|
BMS-466442 |
α adrenergic receptor, IC50: ≥10 μM
|
|
≥98.0% |
Talinolol |
|
Beta-1 adrenergic receptor
|
99.64% |
HOKU-81 |
|
Beta-2 adrenergic receptor
|
|
Nifenalol hydrochloride |
|
|
99.93% |
Desglymidodrine |
α1B-adrenergic receptor, pKi: 5.16
α1A-adrenergic receptor, pKi: 5.89
rat alpha1D-adrenergic receptor, pKi: 5.78
human α2A-adrenoceptor, pKi: 5.83
|
|
|
Metoprolol-d7 hydrochloride |
|
|
99.65% |
Higenamine |
|
|
|
Mibenratide |
|
Beta-1 adrenergic receptor
|
99.77% |
Scopine hydrochloride |
|
|
≥98.0% |
AGN 192836 |
|
|
99.49% |
Bunazosin |
|
|
98.52% |
Efaroxan hydrochloride |
|
|
99.94% |
Prenalterol |
|
|
99.18% |
Salmeterol-d3 |
|
|
98.91% |
CGP 12177 hydrochloride |
|
Beta-2 adrenergic receptor
Beta-1 adrenergic receptor
Beta-3 adrenergic receptor
|
99.57% |
Brombuterol-d9 |
|
|
≥99.0% |
NP10679 |
Alpha-1A adrenergic receptor, IC50: 0.154 μM
Alpha-1A adrenergic receptor, Ki: 0.603 μM
Alpha-2C adrenergic receptor, Ki: 3.09 μM
Alpha-1D adrenergic receptor, Ki: 0.495 μM
Alpha-1B adrenergic receptor, Ki: 1.92 μM
|
|
99.42% |
Amosulalol |
|
Beta-1 adrenergic receptor
|
98.69% |
BMY 14802 |
|
|
98.96% |
Abanoquil |
|
|
98.43% |
(Rac)-Rotigotine hydrochloride |
Alpha-2B adrenergic receptor
|
|
98.66% |
Metoprolol tartrate |
|
|
|
Isoetharine |
|
|
|
Timolol |
|
|
|
Timolol hemihydrate |
|
|
|
(R,R)-Reboxetine mesylate |
|
|
|
Sotalol |
|
|
|
Blonanserin dihydrochloride |
α1-adrenergic receptor, Ki: 26.7 nM
α2-adrenergic receptor, Ki: 530 nM
|
|
|
Doxazosin-d8 |
|
|
|
Rec 15/2615 hydrochloride |
α1B-adrenergic receptor, Ki: 0.3 nM
α1A-adrenergic receptor, Ki: 1.9 nM
Alpha-1D adrenergic receptor, Ki: 2.6 nM
|
|
|
Isamoltane hemifumarate |
|
β-adrenoceptor, IC50: 8.4 nM
|
|
RS-79948-197 |
human α2C-adrenoceptor, Kd: 0.77 nM
rat α2B recepter, Kd: 0.18 nM
rat α2C recepter, Kd: 0.19 nM
human α2A-adrenoceptor, Kd: 0.6 nM
rat α2A receptor, Kd: 0.42 nM
human α2B-adrenoceptor, Kd: 0.46 nM
|
|
|
α1A-AR Degrader 9c |
α1A-adrenergic receptor, DC50: 2.86 μM
|
|
|
Acebutolol |
|
|
|
S(-)-Bisoprolol fumarate |
|
|
|
β2AR agonist /M-receptor antagonist-1 |
|
Beta-2 adrenergic receptor
|
|
Nipradolol |
|
|
|
Agroclavine |
|
|
|
Rezatomidine |
|
|
|
S(-)-Bisoprolol |
|
|
|
Zolertine hydrochloride |
α1B-adrenergic receptor, pKi: 6.81 (in rat liver membrane)
α1A-adrenergic receptor, pKi: 6.35 (in rabbit liver membrane)
|
|
|
Cimbuterol-d9 |
|
|
|
(+)-Sotalol |
|
|
98.82% |
ST91 |
|
|
99.75% |
Ractopamine |
|
pig β2AR, Kd: ~25 nM
pig β1AR, Kd: ~25 nM
|
|
Diacetolol-d7 |
|
|
|
Methyldopate hydrochloride |
|
|
|
Terbutaline sulfate (Standard) |
|
|
|
(±)-Penbutolol-d9 hydrochloride |
|
|
|
Ajmalicine hydrochloride |
α1-adrenergic receptor
α2-adrenergic receptor
|
|
|
BODIPY FL prazosin |
α1B-adrenergic receptor, Ki: 43.3 nM
α1A-adrenergic receptor, Ki: 14.5 nM
|
|
|
Butyryltimolol |
|
|
≥98.0% |
Clozapine (Standard) |
|
|
|
DL 071IT |
|
|
|
Isoprenaline hemisulfate |
|
|
|
Trimazosin |
|
|
|
Phenylethanolamine A-d3 |
|
|
|
AVN-101 hydrochloride |
Alpha-1A adrenergic receptor, Ki: 18.9 nM
Alpha-2A adrenergic receptor, Ki: 1.77 nM
Alpha-2C adrenergic receptor, Ki: 3.55 nM
Alpha-2B adrenergic receptor, Ki: 0.41 nM
Alpha-1D adrenergic receptor, Ki: 30.2 nM
Alpha-1B adrenergic receptor, Ki: 9.4 nM
|
|
|
Asenapine citrate |
α1-adrenergic receptor, pKi: 8.9
Alpha-2A adrenergic receptor, pKi: 8.9
Alpha-2C adrenergic receptor, pKi: 8.9
Alpha-2B adrenergic receptor, pKi: 9.5
|
|
|
JP1302 |
human α2C-adrenoceptor, Ki: 28±2 nM
rodent α2D-adrenoceptor, Ki: 1700±200 nM
human α2A-adrenoceptor, Ki: 3150±50 nM
human α2B-adrenoceptor, Ki: 1470±130 nM
|
|
|
Norepinephrine tartrate |
α1-adrenergic receptor
α2-adrenergic receptor
|
Beta-1 adrenergic receptor
|
|
Fenoterol hydrobromide (Standard) |
|
|
|
β2AR/M3-receptor agonist-1 |
|
β2 adrenoceptor, pEC50: >9.2
|
|
Naftopidil hydrochloride |
Alpha-1A adrenergic receptor, Ki: 3.7 nM
Alpha-1D adrenergic receptor, Ki: 1.2 nM
Alpha-1B adrenergic receptor, Ki: 20 nM
|
|
|
Atenolol (Standard) |
|
Beta-1 adrenergic receptor
|
|
Celiprolol hydrochloride |
|
β adrenergic receptor, Ki: 0.14-8.3 μM
|
|
LAS190792 |
|
β3 adrenoceptor, pIC50: 5.6
β2 adrenoceptor, pIC50: 9.1
β1 adrenoceptor, pIC50: 7.5
|
|
Metoprolol fumarate |
|
|
|
Nifenalol |
|
Beta-1 adrenergic receptor
|
|
Oxyfedrine |
|
|
|
Mabuterol hydrochloride |
|
Beta-2 adrenergic receptor
|
|
Clorprenaline-d7 |
|
|
|
Pronethalol hydrochloride |
|
|
|
Oxprenolol |
|
β-adrenoceptor, Ki: 7.10 nM
|
|
Naftopidil dihydrochloride |
Alpha-1A adrenergic receptor, Ki: 3.7 nM
Alpha-1D adrenergic receptor, Ki: 1.2
Alpha-1B adrenergic receptor, Ki: 20 nM
|
|
|
Meluadrine tartrate |
|
|
|
Bevantolol |
|
Beta-1 adrenergic receptor
|
|
Acebutolol-d7 |
|
|
|
Dapiprazole |
|
|
|
Harmane (Standard) |
|
|
|
Bisoprolol |
|
Beta-1 adrenergic receptor
|
|
Procaterol |
|
|
|
(E)-Guanabenz |
|
|
|
Levobunolol |
|
|
|
Cimaterol |
|
|
|
ST1936 oxalate |
α1-adrenergic receptor, Ki: 390 nM (rat)
α2-adrenergic receptor, Ki: 300 nM (rat)
α2-adrenergic receptor, Ki: 300 nM (human)
|
|
|
Mirtazapine (Standard) |
|
|
|
SB-206606 |
|
Beta-3 adrenergic receptor
|
|
Sulfinalol |
|
|
|
Levobetaxolol |
|
β3 adrenoceptor, IC50: 709 nM
β2 adrenoceptor, IC50: 2970 nM
β1 adrenoceptor, IC50: 33.2 nM
|
|
Celiprolol |
|
β adrenergic receptor, Ki: 0.14-8.3 μM
|
|
Reproterol |
|
|
|
Amidephrine |
|
|
|
Mabuterol |
|
Beta-2 adrenergic receptor
|
|
Bisoprolol fumarate |
|
Beta-1 adrenergic receptor
|
|
Brombuterol-d9 hydrochloride |
|
|
|
TD-5471 hydrochloride |
|
|
|
2-MPMDQ |
α1-adrenergic receptor, Ki: 0.37 nM
α2-adrenergic receptor, Ki: 1740 nM
|
|
|
Bopindolol |
|
β2 adrenoceptor
Beta-1 adrenergic receptor
Beta-3 adrenergic receptor
|
|
4-Hydroxypropranolol-d7 hydrochloride |
|
|
|
Undecylenoyl phenylalanine |
|
|
|
Butaxamine |
|
|
|
BMY 7378 |
rat alpha1D-adrenergic receptor, Ki: 2 nM
rat α1A-adrenergic receptor, Ki: 800 nM
hamster alpha1B-adrenergic receptor, Ki: 600 nM
|
|
|
Bopindolol fumarate |
|
β3 adrenoceptor
β2 adrenoceptor
β1 adrenoceptor
|
|
Mabuterol-d9 |
|
|
|
Xylometazoline |
Alpha-1A adrenergic receptor, Ki: 0.05 μM
Alpha-2A adrenergic receptor, Ki: 0.88 μM
Alpha-2C adrenergic receptor, Ki: 0.19 μM
Alpha-2B adrenergic receptor, Ki: 1.7 μM
Alpha-1D adrenergic receptor, Ki: 0.15 μM
Alpha-1B adrenergic receptor, Ki: 0.30 μM
|
|
|
Meluadrine |
|
|
|
Apraclonidine |
|
|
|
Arformoterol tartrate |
|
Beta-2 adrenergic receptor, Kd: 2.9 nM
|
|
Ecopipam |
Alpha-2A adrenergic receptor, Ki: 731 nM
|
|
|
Moprolol |
|
Beta-1 adrenergic receptor
|
|
Metoprolol-d6 tartrate |
|
|
|
Clenproperol-d7 |
|
|
|
N-5984 |
|
|
|
ARC 239 |
human α2C-adrenoceptor, pKi: 6.95
Alpha-2C adrenergic receptor, pKi: 7.06
|
|
99.71% |
L-Epinephrine sulfate |
|
|
|
Levalbuterol tartrate |
|
|
|
Arformoterol maleate |
|
Beta-2 adrenergic receptor, Kd: 2.9 nM
|
|
Methyldopa hydrochloride |
|
|
|
(rac)-Nebivolol-d4 |
|
|
|
Midodrine |
|
|
99.67% |
Methyldopa |
|
|
|
Pargolol hydrochloride |
|
|
|
Ko-3290 |
|
|
|
LY 344864 hydrochloride |
rat α1-adrenergic receptor, Ki: 5.06 μM
rat α2-adrenergic receptor, Ki: 3.69 μM
|
|
|
Midaglizole hydrochloride |
|
|
99.67% |
Benzquinamide |
|
|
|
Fenmetozole Tosylate |
|
|
|