1. Signaling Pathways
  2. Cell Cycle/DNA Damage
    PI3K/Akt/mTOR
  3. ATM/ATR
  4. ATM/ATR Inhibitors

ATM/ATR Inhibitors

ATM

ATR

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

ATM/ATR Inhibitors & Activators
Product Name ATM ATR Purity
Ceralasertib  
ATR, IC50: 1 nM
99.76%
AZD-7648
ATM, IC50: 17.93 μM
  99.86%
KU-55933
ATM, IC50: 12.9 nM
  99.88%
AZD1390
ATM
  99.28%
KU-60019
ATM, IC50: 6.3 nM
  99.43%
Berzosertib
ATM, Ki: 34 nM
ATR, Ki: 0.2 nM
99.70%
AZD0156
ATM
  99.82%
Elimusertib  
ATR, IC50: 7 nM
99.99%
VE-821
ATM, Ki: 16 μM
ATR, Ki: 13 nM
98.32%
Camonsertib
ATM, IC50: >30 μM
  99.75%
AZ20  
ATR, IC50: 5 nM
99.86%
Elimusertib hydrochloride  
ATR, IC50: 7 nM
99.84%
Gartisertib  
ATR, Ki: <150 pM
99.76%
Lartesertib
ATM
  99.89%
CP-466722
ATM, IC50: 4.1 μM
  99.91%
Ro 90-7501
ATM
  99.10%
AZ32
ATM, IC50: 6.2 nM
ATM, IC50: 0.31 μM (in cell)
  99.94%
CGK733
ATM
ATR
99.83%
Garcinone C  
ATR
99.66%
ETP-46464
ATM, IC50: 545 nM
ATR, IC50: 14 nM
99.55%
NU6027  
ATR
99.04%
AZ31
ATM, IC50: 1.2 nM
ATM, IC50: 46 nM (in cell)
  98.13%
ATR-IN-19  
ATR
ATR-IN-15
ATM, IC50: > 10000 nM
ATR, IC50: 8 nM
ATM Inhibitor-4
ATM, IC50: 0.32 nM
 
Abd110  
ATR
ATR-IN-16  
ATR
ATR-IN-29  
ATR, IC50: 1 nM
ATR-IN-14  
ATR
ATR-IN-10  
ATR, IC50: 2.978 μM
A011
ATM, IC50: 1.0 nM
 
ATR-IN-17  
ATR
ATM Inhibitor-2
ATM, IC50: <1 nM
 
ATR-IN-21  
ATR, IC50: <1000 nM
ATR-IN-20
ATM, IC50: 100 nM
ATR, IC50: 3 nM
ATR-IN-13  
ATR, IC50: 2 nM
ATR-IN-18  
ATR, IC50: 0.69 nM
Antitumor agent-28
ATM
ATR
ATM Inhibitor-3
ATM, IC50: 0.71 nM
 
ATM Inhibitor-1
ATM, IC50: 0.7 nM
ATM, IC50: 2.8 nM (Cellular assay)