1. Signaling Pathways
  2. GPCR/G Protein
  3. P2Y Receptor
  4. P2Y Receptor Inhibitors

P2Y Receptor Inhibitors

P2Y1 Receptor

P2Y2 Receptor

P2Y6 Receptor

P2Y12 Receptor

P2Y13 Receptor

P2Y14 Receptor

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

P2Y Receptor Inhibitors, Agonists, Antagonists, Activators & Modulators
Product Name P2Y1 Receptor P2Y2 Receptor P2Y6 Receptor P2Y12 Receptor P2Y13 Receptor P2Y14 Receptor Purity
Ticagrelor      
P2Y12 Receptor
    99.95%
Clopidogrel      
P2Y12 Receptor
    99.57%
Uridine 5′-diphosphoglucose disodium          
P2Y14 Receptor
99.98%
P2Y14R antagonist 3          
P2Y14 Receptor, IC50: 23.6 nM
P2Y14 Receptor, Kd: 7.26 μM
UDP-Galactose disodium          
P2Y14 Receptor, EC50: 0.67 μM
99.42%
Cangrelor tetrasodium      
P2Y12 Receptor
    99.96%
Diquafosol tetrasodium  
P2Y2 Receptor
        ≥99.0%
MRS 2578    
P2Y6 Receptor
      98.15%
Uridine-5'-diphosphate disodium salt    
P2Y6 Receptor
      99.23%
YM-254890
P2Y1 Receptor
          ≥99.0%
AR-C118925XX  
P2Y2 Receptor
        ≥99.0%
PSB-0739      
P2Y12 Receptor
    ≥98.0%
Clopidogrel hydrogen sulfate      
P2Y12 Receptor
    99.88%
PPTN hydrochloride          
P2Y14 Receptor
99.89%
2-MeS-ADP trisodium      
P2Y12 Receptor
P2Y13 Receptor
  99.90%
BPTU
P2Y1 Receptor
          99.67%
Prasugrel      
P2Y12 Receptor
    99.85%
MRS2500 tetraammonium
P2Y1 Receptor
          99.85%
Uridine 5′-diphosphoglucose (Standard)          
P2Y14 Receptor
Prasugrel hydrochloride      
P2Y12 Receptor
    98.49%
2-Methylthio-AMP      
P2Y12 Receptor
    98.94%
PIT
P2Y1 Receptor, IC50: 0.14 μM μM
          99.07%
AZD1283      
P2Y12 Receptor, IC50: 11 nM
    99.33%
Clopidogrel thiolactone      
P2Y12 Receptor
    ≥98.0%
ADP-β-S trilithium      
P2Y12 Receptor
   
P2Y6R antagonist 1    
P2Y6 Receptor, IC50: 19.6 nM
      99.94%
Elinogrel      
P2Y12 Receptor
    98.68%
P2Y14R antagonist 2          
P2Y14 Receptor, IC50: 0.40 nM
99.56%
4-Thiouridine 5′-triphosphate tetralithium  
P2Y2 Receptor, EC50: 35 nM
       
MRS2768 tetrasodium salt  
P2Y2 Receptor
        98.70%
P2Y14R antagonist 1
P2Y1 Receptor, IC50: > 100 nM
P2Y2 Receptor, IC50: > 100 nM
P2Y6 Receptor, IC50: 89.7 nM
P2Y12 Receptor, IC50: > 100 nM
 
P2Y14 Receptor, IC50: 0.6 nM
98.58%
MRS2365
P2Y1 Receptor, EC50: 0.4 nM
         
Ticagrelor-d7      
P2Y12 Receptor
   
MRS2365 trisodium
P2Y1 Receptor, EC50: 0.4 nM
          ≥99.0%
MRS2279 diammonium
P2Y1 Receptor, IC50: 51.6 nM
          ≥98.0%
Prasugrel-d3      
P2Y12 Receptor
    98.58%
2-Methylthio-AMP diTEA      
P2Y12 Receptor
    ≥98.0%
Adenosine 2',5'-diphosphate sodium
P2Y1 Receptor
          ≥99.0%
Uridine 5′-diphosphoglucose          
P2Y14 Receptor
Cangrelor      
P2Y12 Receptor
   
SAR216471 hydrochloride      
P2Y12 Receptor
   
P2Y1/P2Y6 antagonist 1
P2Y1 Receptor, IC50: 9.72 μM
 
P2Y6 Receptor, IC50: 1.89 μM
     
Uridine 5'-O-thiodiphosphate trisodium    
P2Y6 Receptor, EC50: 28 nM
     
HDL-16          
P2Y14 Receptor, IC50: 0.3095 nM
99.19%
UDP-Galactose          
P2Y14 Receptor, EC50: 0.67 μM
Diquafosol  
P2Y2 Receptor
       
Regrelor disodium      
P2Y12 Receptor
   
4-Thiouridine 5′-triphosphate tetrasodium  
P2Y2 Receptor, EC50: 35 nM
       
P2Y14R antagonist 4          
P2Y14 Receptor, IC50: 5.6 nM
P2Y14R antagonist 5          
P2Y14 Receptor, IC50: 23.60 nM
Prasugrel-d5      
P2Y12 Receptor
   
MRS-2179
P2Y1 Receptor
         
TNP-ATP tetrasodium
P2Y1 Receptor, IC50: 6 nM
         
2-MeSADP      
P2Y12 Receptor, EC50: 5 nM
P2Y13 Receptor, EC50: 19 nM
 
Blue FPG-A trisodium
P2Y1 Receptor, IC50: 2.6 μM
         
MRS2693 ammonium    
P2Y6 Receptor, EC50: 0.015 μM
     
MRS2279
P2Y1 Receptor, IC50: 51.6 nM
         
MRS4833          
hP2Y14R, IC50: 5.92 nM
mP2Y14R, IC50: 4.8 nM
5-OMe-UDP    
P2Y6 Receptor, EC50: 0.08 μM
     
Uridine 5′-diphosphoglucose-13C disodium    
P2Y6 Receptor
     
MRS2496
P2Y1 Receptor
         
P2Y1 antagonist 1
P2Y1 Receptor
         
Sp-UTP-α-S  
P2Y2 Receptor
       
MRS2905 trisodium          
P2Y14 Receptor, EC50: 0.92 nM
Prasugrel (Maleic acid)      
P2Y12 Receptor
   
UDP-GlcNAc          
P2Y14 Receptor
MRS2603
P2Y1 Receptor
     
P2Y13 Receptor
 
Elinogrel potassium      
P2Y12 Receptor
   
(Rac)-BX 048      
P2Y12 Receptor
   
2-Thio-UTP  
P2Y2 Receptor, EC50: 50 nM