1. Signaling Pathways
  2. Stem Cell/Wnt
    TGF-beta/Smad
  3. PKA
  4. PKA Inhibitors

PKA Inhibitors

PKA

PKAR

PKACα

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

PKA Inhibitors, Agonists & Activators
Product Name PKA PKAR PKACα Purity
Bucladesine sodium
PKA
    99.48%
PKC-IN-6
PKA, IC50: >500 μM
    99.63%
Fasudil Hydrochloride
PKA, IC50: 4.58 μM
    99.97%
Bucladesine calcium
PKA
    98.63%
Daphnetin
PKA, IC50: 9.33 μM
    99.77%
KT5823
PKA, Ki: 10 μM
    99.90%
AT7867
PKA, IC50: 20 nM
    99.88%
Bilobetin
PKA
    99.39%
PKA Inhibitor Fragment (6-22) amide TFA
PKA, Ki: 2.8 nM
    99.87%
AT13148
PKA, IC50: 3 nM
    99.20%
CW 008
PKA
    98.15%
AT7867 dihydrochloride
PKA, IC50: 20 nM
    99.75%
Sp-cAMPS sodium salt
PKA I
PKA II
    99.45%
Hu7691
PKA, IC50: 11 nM
    99.91%
Jaspamycin
Trypanosoma brucei PKA holoenzyme, Kd: 8 nM
Trypanosoma brucei PKAR(199-499), EC50: 6.5 nM
  98.60%
Undecane
PKA
    99.66%
A-3 hydrochloride
PKA, Ki: 4.3 μM
    99.75%
PF-4950834
PKA, IC50: 424 nM
    99.60%
Sp-cAMPS
PKA I
PKA II
   
Akt1&PKA-IN-1
PKAa, IC50: 0.03 μM
   
Fasudil
PKA, IC50: 4.58 μM
   
Hu7691 free base
PKA, IC50: 11 nM
   
Fasudil hydrochloride semihydrate
PKA, IC50: 4.58 μM
   
Fasudil dihydrochloride
PKA, IC50: 4.58 μM
    99.98%
Sp-8-Br-cAMPS sodium
PKA, EC50: 360 nM
   
GSK-3α/β-IN-1
PKA, IC50: 0.188 μM
   
Sp-cAMPS triethylamine
PKA I
PKA II
   
PKA Inhibitor Fragment (6-22) amide
PKA, Ki: 2.8 nM
   
HA-100 dihydrochloride
PKA, IC50: 8 μM
   
GSK466317A
PKA, IC50: 12.59 μM
   
HA-100 hydrochloride
PKA, IC50: 8 μM
   
PKA-IN-2    
J-PKACα, IC50: 6.3 nM
LX7101 monohydrochloride
PKA, IC50: <1 nM
   
Balanol
PKA