1. Signaling Pathways
  2. Membrane Transporter/Ion Channel
  3. GLUT
  4. GLUT Inhibitors

GLUT Inhibitors

GLUT1

GLUT2

GLUT3

GLUT4

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

GLUT Inhibitors & Activators
Product Name GLUT1 GLUT2 GLUT3 GLUT4 Purity
BAY-876
GLUT1, IC50: 2 nM
GLUT2, IC50: 10.08 μM
GLUT3, IC50: 1.67 μM
GLUT4, IC50: 0.29 μM
98.46%
Phloretin
GLUT1
GLUT2
    99.67%
WZB117
GLUT1
      99.97%
KL-11743
GLUT1, IC50: 115 nM
GLUT2, IC50: 137 nM
GLUT3, IC50: 90 nM
GLUT4, IC50: 68 nM
98.80%
STF-31
GLUT1, IC50: 1 μM
      98.01%
Avicularin (Standard)      
GLUT4
Phloretin (Standard)
GLUT1
GLUT2
   
Rhoifolin      
GLUT4
99.09%
MOTS-c(human) acetate      
GLUT4
98.97%
Fasentin      
GLUT4, IC50: 68 μM
≥98.0%
Avicularin      
GLUT4
99.48%
GLUT inhibitor-1
GLUT1, IC50: 242 nM
 
GLUT3, IC50: 179 nM
  98.01%
Licarin B      
GLUT4
99.93%
GLUT4 activator 1      
GLUT4, EC50: 0.14 μM
99.71%
GLUT4-IN-2
GLUT1, IC50: 11.4 μM
   
GLUT4, IC50: 6.8 μM
99.90%
4,6-O-Ethylidene-α-D-glucose
GLUT1
      ≥98.0%
Lavendustin B
GLUT1, Ki: 15 μM
      98.04%
Sennidin B      
GLUT4
98.83%
GLUT1-IN-1
GLUT1
     
Sennidin A      
GLUT4