2. GPCR/G Protein
  3. GCGR
  4. DA-302168S

DA-302168S 是一种口服有效的选择性 GLP-1R 激动剂，其 EC50 值为 1.32 nM。DA-302168S 可刺激胰岛素分泌，并具有降血糖作用。DA-302168S 可减少食物摄入量。DA-302168S 主要激活猴和人的 GLP-1R，对大鼠、小鼠和犬的 GLP-1R 几乎无激动作用。DA-302168S 可用于 2 型糖尿病和肥胖症研究。

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DA-302168S

DA-302168S Chemical Structure

CAS No. : 2969158-02-7

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DA-302168S 相关抗体

Top Publications Citing Use of Products

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

DA-302168S is an orally active and selective agonist targeting the GLP-1R, with EC50 value of 1.32 nM. DA-302168S stimulates insulin secretion and shows hypoglycemic effects. DA-302168S decreases food intake. DA-302168S mainly activates GLP-1R of monkeys and humans, and exhibits little excitatory effect on GLP-1R of rats, mice, and dogs. DA-302168S can be used for type 2 diabetes and obesity study[1].

Clinical Trial
分子量

616.01

Formula

C33H24ClF2N3O5
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

DA-302168S 相关分类

  • 摩尔计算器

  • 稀释计算器

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

DA-302168S2969158-02-7GCGRGlucagon ReceptorhypoglycemicHEK293 cellsInhibitorinhibitorinhibit

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产品名称：
DA-302168S
目录号：
HY-172811
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