2. Metabolic Enzyme/Protease
  3. Dipeptidyl Peptidase
  4. 5-Hydroxy saxagliptin hydrochloride

5-Hydroxy saxagliptin hydrochloride  (Synonyms: 5-羟基沙格列汀 (盐酸盐))

目录号: HY-W741755A
产品使用指南 技术支持

5-Hydroxy saxagliptin hydrochloride 是 Saxagliptin (HY-10285) 的活性代谢产物，也是一种强效的和选择性的 DPP-4 抑制剂。5-Hydroxy saxagliptin hydrochloride 对人和食蟹猴的 Ki 值分别为 2.6 nM 和 2.9 nM。5-Hydroxy saxagliptin hydrochloride 可用于2 型糖尿病的研究。

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5-Hydroxy saxagliptin hydrochloride

5-Hydroxy saxagliptin hydrochloride Chemical Structure

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5-Hydroxy saxagliptin hydrochloride 相关抗体

Top Publications Citing Use of Products

查看 Dipeptidyl Peptidase 亚型特异性产品:

查看所有亚型
DPP-1 DPP-2 DPP-4 DPP-8 DPP-9

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

5-Hydroxy saxagliptin hydrochloride is an active metabolite of Saxagliptin (HY-10285) and a potent and selective DPP-4 inhibitor. 5-Hydroxy saxagliptin hydrochloride has Ki values of 2.6 nM and 2.9 nM for humans and cynomolgus monkeys, respectively. 5-Hydroxy saxagliptin hydrochloride can be used in the research of type 2 diabetes mellitus[1].

IC50 & Target[1]

DPP-4

2.6 nM (Ki)

DPP-8

2495 nM (Ki)

DPP-9

423 nM (Ki)

分子量

367.87

Formula

C18H26ClN3O3
中文名称

5-羟基沙格列汀 (盐酸盐)
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

5-Hydroxy saxagliptin hydrochloride 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

5-Hydroxy saxagliptin5-羟基沙格列汀 (盐酸盐)Dipeptidyl PeptidaseDPPSaxagliptincynomolgus monkeystype 2 diabetes mellitusInhibitorinhibitorinhibit

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