1. GPCR/G Protein
  2. GNRH Receptor
  3. Cetrorelix diacetate

Cetrorelix diacetate (Synonyms: SB-75 diacetate)

目录号: HY-P0009B
产品使用指南

Cetrorelix diacetate (SB-075 diacetate)是 GnRH 受体的强效拮抗剂,其 IC50 值为 1.21 nM。

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Cetrorelix diacetate Chemical Structure

Cetrorelix diacetate Chemical Structure

CAS No. : 130143-01-0

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Cetrorelix diacetate 的其他形式现货产品:

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Description

Cetrorelix diacetate (SB-075 diacetate) is a potent gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM[1].

IC50 & Target

IC50: 1.21 nM GnRH[1].

In Vitro

Cetrorelix diacetate inhibits growth of ES-2 cell line at 1000 ng/ml. Cetrorelix diacetate has comparable antiproliferative effects as GnRH-I agonists indicating that the dichotomy of GnRH-I agonists and antagonists might not apply to the GnRH-I system in cancer cells[2].

Molecular Weight

1551.14

Formula

C₇₄H₁₀₀ClN₁₇O₁₈

CAS No.

130143-01-0

Sequence Shortening

Ac-{2-Naph-Ala}-{Cl-Phe}-{3Py-Ala}-SY-{Cit}-LRPA-NH2

中文名称

二醋酸西曲瑞克

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Keywords:

Cetrorelix diacetateSB-75 diacetateGNRH ReceptorGonadotropin releasing hormone receptorGNRHRInhibitorinhibitorinhibit

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产品名称:
Cetrorelix diacetate
目录号:
HY-P0009B
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