2. GPCR/G Protein Neuronal Signaling
  3. 5-HT Receptor
  4. CP-135807

CP-135807 是一种口服有效、选择性的 5-HT1D 激动剂 (IC50=3.1 nM)。CP-135807 介导中枢精神活性，可用于抗抑郁研究。

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CP-135807 Chemical Structure

CP-135807 Chemical Structure

CAS No. : 151272-90-1

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规格 价格 是否有货
5 mg ￥2331
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Customer Review

CP-135807 相关抗体

Top Publications Citing Use of Products

查看 5-HT Receptor 亚型特异性产品:

查看所有亚型
5-HT1 Receptor 5-HT2 Receptor 5-HT3 Receptor 5-HT4 Receptor 5-HT5 Receptor 5-HT6 Receptor 5-HT7 Receptor 5-HT Receptor

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

CP-135807 is an orally active and selective 5-HT1D agonist (IC50=3.1 nM), bovine). CP-135807 mediates central psychoactivity and can be used in antidepressant research[1][2].

IC50 & Target[1][2]

5-HT1D Receptor

3.1 nM (IC50, rat)

5-HT1D Receptor

33 nM (IC50, bovine)

体内研究
(In Vivo)

鸽子被训练在一个固定比例的食物提供下啄一个键。CP-135807 (0.1 mg/kg; 肌肉注射; 单剂量) 则能够完全和剂量依赖地替代成年雄性卡诺鸽子的训练剂量[1]。

MCE has not independently confirmed the accuracy of these methods. They are for reference only.
分子量

351.40

Formula

C19H21N5O2
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

CP-135807 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

CP-135807151272-90-1CP135807CP 1358075-HT ReceptorSerotonin Receptor5-hydroxytryptamine ReceptorInhibitorinhibitorinhibit

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产品名称：
CP-135807
目录号：
HY-103092
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