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  4. hCES2A-IN-1

hCES2A-IN-1 (compound 20w) 是一种有效的 hCES2A 抑制剂，IC50 值为 1.6 nM。 hCES2A-IN-1 是一种 bysspectin A 衍生物，与先导化合物 bysspectin A 相比，性能提高了约 1000 倍。

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hCES2A-IN-1 Chemical Structure

hCES2A-IN-1 Chemical Structure

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hCES2A-IN-1 相关抗体

Top Publications Citing Use of Products

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

hCES2A-IN-1 (compound 20w) is a potent hCES2A inhibitor, with an IC50 value of 1.6 nM. hCES2A-IN-1, a bysspectin A derivative, shows an approximately 1000-fold improvement over the lead compound bysspectin A[1].

IC50 & Target

hCES2A (0.0016 ± 0.00034 μM), hCES1A (7.26 ± 0.94 μM)[1]
体外研究
(In Vitro)

hCES2A-IN-1 (compound 20w) 在浓度低于 10 μM 时对 HepG2 细胞表现出非常弱的细胞毒性[1]。
hCES2A-IN-1 能够以剂量依赖性方式抑制活细胞中 hCES2A 介导的 NCEN 水解，IC50 值为 0.052 μM，其抑制活性显着高于 Loperamide，IC50 值为 1.44 μM[1]。
hCES2A-IN-1 表现出良好的代谢稳定性，在人肝微粒体I相或II相代谢系统中的半衰期分别为125.96分钟和97.38分钟[1]。

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

hCES2A-IN-1 相关抗体:
分子量

366.45

Formula

C23H26O4
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

hCES2A-IN-1 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

hCES2A-IN-1OthersInhibitorinhibitorinhibit

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