2. Membrane Transporter/Ion Channel
  3. Sodium Channel
  4. Pilsicainide

Pilsicainide  (Synonyms: SUN 1165 free base; Pilzicainide)

目录号: HY-133715
产品使用指南

摩尔计算器

Pilsicainide (SUN 1165 free acid) 是一种有效的钠通道 (sodium channel) 阻滞剂和有效的 Ic 类抗心律失常剂。

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Pilsicainide Chemical Structure

Pilsicainide Chemical Structure

CAS No. : 88069-67-4

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Pilsicainide 的其他形式现货产品:

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Other Forms of Pilsicainide:

Pilsicainide 相关抗体

Top Publications Citing Use of Products

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

Pilsicainide (SUN 1165 free acid) is a potent sodium channel blocker and potent class Ic antiarrhythmic agent[1][2].

体外研究
(In Vitro)

Pilsicainide (SUN 1165 free acid; 10-200 μg/mL) decreases peak amplitude of the net inward current in a dose-dependent manner with an IC50 of 29.2 μg/mL in levo-thyroxine (T4)-treated rat atrial cells[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Pilsicainide 相关抗体:
体内研究
(In Vivo)

Pilsicainide (SUN 1165 free acid; 2 mg/kg; i.v.; once) decreases the conduction velocity in T4-treated rat atrium by decreasing the Max dV/dt and net inward current[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model: Male Sprague-Dawley (SD) rats weighing from 200 to 220 g, with levo-thyroxine (T4) treatment[1]
Dosage: 2 mg/kg
Administration: Bolus injection into right external carotid vein within 2 minutes, once
Result: Elongated the QT interval at 15 and 60 minutes after administration.
Shortened P wave and QRS complex durations.
Markedly decreased action potential amplitudes (APA) and Max dV/dt, and significantly lengthened the action potential durations.
Clinical Trial
分子量

272.39

Formula

C17H24N2O
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

Pilsicainide 相关分类

  • 摩尔计算器

  • 稀释计算器

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  • Do most proteins show cross-species activity?

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Keywords:

Pilsicainide88069-67-4SUN 1165 PilzicainideSUN1165SUN-1165Sodium ChannelNa channelsNa+ channelsatrial tachyarrhythmiasantiarrhythmicorally activeInhibitorinhibitorinhibit

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