2. Metabolic Enzyme/Protease
  3. Phosphodiesterase (PDE)
  4. Deltasonamide 2

Deltasonamide 2 是一种竞争性的，高亲和力的 PDEδ 抑制剂，Kd 值约为 385 pM。

在相同的摩尔浓度下，化合物盐形式与游离形式有相同的生物活性，但盐形式 Deltasonamide 2 (TFA) 和 Deltasonamide 2 hydrochloride 通常具有更好的水溶性和稳定性。

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Deltasonamide 2

Deltasonamide 2 Chemical Structure

CAS No. : 2088485-34-9

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Deltasonamide 2 的其他形式现货产品:

Customer Review

Other Forms of Deltasonamide 2:

Deltasonamide 2 相关抗体

Top Publications Citing Use of Products

MCE 顾客使用本产品发表的 1 篇科研文献

查看 Phosphodiesterase (PDE) 亚型特异性产品:

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PDE1 PDE2 PDE3 PDE4 PDE5 PDE6 PDE7 PDE9 PDE10 PDE11 PDE12 PDE8 Autotaxin

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

Deltasonamide 2 is a competitive, high affinity PDEδ inhibitor with a Kd of ~385 pM[1].

IC50 & Target

Kd: ~385 pM (PDEδ)[1]
细胞效力
(Cellular Effect)
Cell Line Type Value Description References
AGS IC50
1.2 μM
Compound: Deltasonamide 2
Antiproliferative activity against human AGS cells assessed as reduction in cell viability measured after 3 days by Celltiter-Glo assay
Antiproliferative activity against human AGS cells assessed as reduction in cell viability measured after 3 days by Celltiter-Glo assay
[PMID: 34965125]
MIA PaCa-2 IC50
507 nM
Compound: Deltasonamide 2
Antiproliferative activity against human MIA PaCa-2 cells assessed as reduction in cell viability measured after 3 days by Celltiter-Glo assay
Antiproliferative activity against human MIA PaCa-2 cells assessed as reduction in cell viability measured after 3 days by Celltiter-Glo assay
[PMID: 34965125]
NCI-H358 IC50
954 nM
Compound: Deltasonamide 2
Antiproliferative activity against human NCI-H358 cells assessed as reduction in cell viability measured after 3 days by Celltiter-Glo assay
Antiproliferative activity against human NCI-H358 cells assessed as reduction in cell viability measured after 3 days by Celltiter-Glo assay
[PMID: 34965125]
PaTu 8988t IC50
1.2 μM
Compound: Deltasonamide 2
Antiproliferative activity against human PaTu 8988t cells assessed as reduction in cell viability measured after 3 days by Celltiter-Glo assay
Antiproliferative activity against human PaTu 8988t cells assessed as reduction in cell viability measured after 3 days by Celltiter-Glo assay
[PMID: 34965125]
分子量

647.25

Formula

C30H39ClN6O4S2
CAS 号
性状

固体

颜色

White to off-white

运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

Deltasonamide 2 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Deltasonamide 22088485-34-9Deltasonamide2Deltasonamide-2Phosphodiesterase (PDE)Inhibitorinhibitorinhibit

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目录号：
HY-122641A
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