1. GPCR/G Protein Neuronal Signaling
  2. Neurokinin Receptor
  3. MEN 10207 acetate

MEN 10207 (acetate) 是一种 NK-2 速激肽受体的选择性拮抗剂。MEN 10207 (acetate) 可引起大鼠膀胱和豚鼠气道体内速激肽诱导的收缩。MEN 10207 (acetate) 可抑制 [β-Ala 8]-NKA (4-10) 诱导的麻醉大鼠膀胱运动增强,以及 [β-Ala 8]-NKA (4-10) 诱导的麻醉豚鼠支气管收缩增强。

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Custom Peptide Synthesis

MEN 10207 acetate

MEN 10207 acetate Chemical Structure

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MEN 10207 acetate 的其他形式现货产品:

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Other Forms of MEN 10207 acetate:

MCE 顾客使用本产品发表的 1 篇科研文献

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生物活性

MEN 10207 (acetate) is a selective antagonist of the NK-2 tachykinin receptor. MEN 10207 (acetate) induces tachykinin-induced contractions in rat bladder and guinea pig airways in vivo. MEN 10207 (acetate) inhibits [β-Ala 8 ]-NKA (4-10)-induced enhancement of bladder motility in anesthetized rats and [β-Ala 8 ]-NKA (4-10)-induced enhancement of bronchoconstriction in anesthetized guinea pigs[1].

IC50 & Target[1]

NK2R

 

分子量

1109.24

Formula

C57H68N14O10.xC2H4O2

Sequence

Asp-Tyr-{d-Trp}-Val-{d-Trp}-{d-Trp}-Arg

Sequence Shortening

DY-{d-Trp}-V-{d-Trp}-{d-Trp}-R

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.

纯度 & 产品资料
参考文献
  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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产品名称:
MEN 10207 acetate
目录号:
HY-151413A
需求量: