2. Epigenetics
  3. Epigenetic Reader Domain
  4. PBRM1-BD2-IN-6

PBRM1-BD2-IN-6 是一种有效的 PBRM1 溴区结构域抑制剂，IC50 值为 0.22 µM。PBRM1-BD2-IN-6 显示出抗增殖活性。PBRM1-BD2-IN-6 具有研究 PBRM1 依赖性癌症的潜力。

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PBRM1-BD2-IN-6 Chemical Structure

PBRM1-BD2-IN-6 Chemical Structure

CAS No. : 2819989-67-6

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PBRM1-BD2-IN-6 相关抗体

Top Publications Citing Use of Products

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

PBRM1-BD2-IN-6 is a potent PBRM1 bromodomain inhibitor with an IC50 value of 0.22 µM. PBRM1-BD2-IN-6 shows antiproliferation activity. PBRM1-BD2-IN-6 has the potential for the research of PBRM1-dependent cancer[1].

IC50 & Target

IC50: 0.22 nM (PBRM1-BD2)[1]
体外研究
(In Vitro)

PBRM1-BD2-IN-6 (compound 25) (0.1, 1, 10 μM; 5 days) shows antiproliferation activity with IC50 values of 0.66, 0.77, 0.32 µM for LNCaP, PC3, HEK293T cells, respectively[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

PBRM1-BD2-IN-6 相关抗体:

Cell Proliferation Assay[1]

Cell Line: LNCaP, PC3, HEK293T cells
Concentration: 0.1, 1, 10 μM
Incubation Time: 5 days
Result: Inhibited the cell growth with IC50 values of 0.66, 0.77, 0.32 µM for LNCaP, PC3, HEK293T cells, respectively.
分子量

286.76

Formula

C16H15ClN2O
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

PBRM1-BD2-IN-6 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

PBRM1-BD2-IN-62819989-67-6Epigenetic Reader DomainantiproliferationLNCaPPC3HEK293T cellscancerInhibitorinhibitorinhibit

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目录号：
HY-151533
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