2. Others Neuronal Signaling GPCR/G Protein
  3. 5-HT Receptor Isotope-Labeled Compounds
  4. Sarpogrelate-d4 hydrochloride

Sarpogrelate-d4 hydrochloride  (Synonyms: 盐酸沙格雷酯-d4; MCI-9042-d4)

目录号: HY-10564S1
产品使用指南 技术支持

Sarpogrelate-d4 (MCI-9042-d4) hydrochloride 是氘代标记的 Sarpogrelate (hydrochloride)。Sarpogrelate hydrochloride (MCI-9042) 是一种选择性的 5-HT2R 拮抗剂，对 5-HT2A，5-HT2B，和 5-HT2C 受体的 pKi 值分别为 8.52、6.57 和 7.43。Sarpogrelate hydrochloride 对 5-HT1，5-HT3，5-HT4，α1-，α2- 和 β-肾上腺素受体，组胺 H1，H2 以及毒蕈碱 M3 受体缺乏显著的拮抗活性。Sarpogrelate hydrochloride 可用于研究与血栓形成有关的血管疾病。

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Sarpogrelate-d<sub>4</sub> hydrochloride Chemical Structure

Sarpogrelate-d4 hydrochloride Chemical Structure

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Other Forms of Sarpogrelate-d4 hydrochloride:

Sarpogrelate-d4 hydrochloride 相关抗体

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  • 生物活性

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生物活性

Sarpogrelate-d4 (MCI-9042-d4) hydrochloride is deuterium labeled Sarpogrelate (hydrochloride). Sarpogrelate hydrochloride (MCI-9042) is a selective 5-HT2R antagonist, with pKis of 8.52, 6.57, and 7.43 for 5-HT2A, 5-HT2B, and 5-HT2C receptors, respectively. Sarpogrelate hydrochloride displays selectivity over 5-HT1, 5-HT3, 5-HT4, α1-, α2- and β-adrenoreceptor, histamine H1, H2 and muscarinic M3 receptors. Sarpogrelate hydrochloride can be used for the research of vascular disease associated with thrombosis[1][2][3][4].

IC50 & Target

5-HT2A Receptor

 

5-HT2B Receptor

 

5-HT2C Receptor

 

分子量

469.99

同用名

盐酸沙格雷酯-d4; MCI-9042-d4

Formula

C24H28D4ClNO6
非标记 CAS
中文名称

盐酸沙格雷酯-d4；沙格雷酯盐酸盐-d4
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

Sarpogrelate-d4 hydrochloride 相关分类

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The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Sarpogrelate-d4MCI-9042-d4盐酸沙格雷酯-d4沙格雷酯盐酸盐-d45-HT ReceptorIsotope-Labeled CompoundsSerotonin Receptor5-hydroxytryptamine ReceptorInhibitorinhibitorinhibit

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