2. Metabolic Enzyme/Protease
  3. UGT
  4. UGT1A1-IN-1

UGT1A1-IN-1 (compound 2) 是非竞争性 UGT1A1 抑制剂，能够抑制 UGT1A1 介导的 1-O-葡糖苷酸化过程，其 Ki 值为 5.02 μM。UGT1A1-IN-1 可以与 UGT1A1 结合在与胆红素 (HY-N0323) 相同的配体结合位点上。UGT1A1-IN-1 可以作为 UGT1A1 的“开启”荧光探针底物。

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UGT1A1-IN-1 Chemical Structure

UGT1A1-IN-1 Chemical Structure

CAS No. : 2097024-37-6

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UGT1A1-IN-1 相关抗体

Top Publications Citing Use of Products

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

UGT1A1-IN-1 (compound 2) is a non-competitive inhibitor of UGT1A1, which can inhibit the 1-O-glucuronidation process mediated by UGT1A1 with a Ki value of 5.02 μM. UGT1A1-IN-1 (compound 2) can bind on UGT1A1 at the same ligand-binding site as bilirubin (HY-N0323). UGT1A1-IN-1 can serve as a ‘turn-on’ fluorescent probe substrate for UGT1A1[1].

IC50 & Target

Ki: 5.02 μM (UGT1A1)[1].
分子量

345.39

Formula

C22H19NO3
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

UGT1A1-IN-1 相关分类

  • 摩尔计算器

  • 稀释计算器

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  • Do most proteins show cross-species activity?

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Keywords:

UGT1A1-IN-12097024-37-6UGTUDP-glucuronosyltransferaseUridine diphosphate glucuronosyltransferaseprobemetabolic diseaseInhibitorinhibitorinhibit

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产品名称：
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目录号：
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