1. GPCR/G Protein Neuronal Signaling
  2. Opioid Receptor
  3. AT-121 hydrochloride

AT-121 hydrochloride 是一种双功能的 nociception 和 mu 阿片受体 (mu opioid receptor) 激动剂,Ki 值分别为 3.67 和 16.49 nM。AT-121 hydrochloride 是一种安全、无成瘾性的缓解疼痛化合物,具有抗伤害和止痛作用。

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AT-121 hydrochloride Chemical Structure

AT-121 hydrochloride Chemical Structure

CAS No. : 2099681-71-5

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  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

AT-121 hydrochloride is a bifunctional nociception and mu opioid receptor agonist, with Kis of 3.67 and 16.49 nM, respectively. AT-121 hydrochloride is a safe, non-addictive analgesic, and shows antinociceptive and antiallodynic effects[1].

体内研究
(In Vivo)

AT-121 hydrochloride (0.003-0.03 mg/kg; s.c.) produces potent antinociceptive effect[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model: Adult male and female rhesus monkeys[1]
Dosage: 0.003-0.03 mg/kg
Administration: Subcutaneous
Result: Produced antinociceptive effects against an acute noxious stimulus, 50 °C water, in a dose-dependent.
分子量

499.11

Formula

C24H39ClN4O3S

CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.

纯度 & 产品资料
参考文献

AT-121 hydrochloride 相关分类

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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产品名称:
AT-121 hydrochloride
目录号:
HY-112692A
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