1. GPCR/G Protein Neuronal Signaling
  2. Opioid Receptor
  3. AT-121

AT-121 是一种双功能的 nociception 和 mu 阿片受体 (mu opioid receptor) 激动剂,Ki 值分别为 3.67 和 16.49 nM。AT-121 是一种安全、无成瘾性的缓解疼痛药,具有抗伤害和止痛作用。

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AT-121 Chemical Structure

AT-121 Chemical Structure

CAS No. : 2099681-31-7

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100 μg(2.16 mM * 100 μL in Chloroform) ¥1480
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生物活性

AT-121 is a bifunctional nociception and mu opioid receptor agonist, with Kis of 3.67 and 16.49 nM, respectively. AT-121 is a safe, non-addictive analgesic, and shows antinociceptive and antiallodynic effects[1].

体内研究
(In Vivo)

AT-121 (0.003-0.03 mg/kg; s.c.) produces potent antinociceptive effect[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model: Adult male and female rhesus monkeys[1]
Dosage: 0.003-0.03 mg/kg
Administration: Subcutaneous
Result: Produced antinociceptive effects against an acute noxious stimulus, 50 °C water, in a dose-dependent.
分子量

462.65

Formula

C24H38N4O3S

CAS 号
性状

液体

颜色

Colorless to light yellow

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Solution, -20°C, 2 years

纯度 & 产品资料

纯度: ≥96.0%

参考文献
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产品名称:
AT-121
目录号:
HY-112692
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