2. GPCR/G Protein Neuronal Signaling Immunology/Inflammation
  3. Histamine Receptor
  4. GT-2016

GT-2016 是一种有效的、选择性的可穿过血脑屏障的组胺 H3 受体拮抗剂，Ki 为 43.8 nM。GT-2016 对 H1 和 H2 受体具有选择性，并对组胺甲基转移酶无活性。

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GT-2016 Chemical Structure

GT-2016 Chemical Structure

CAS No. : 152241-24-2

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规格 价格 是否有货
1 mg ￥666
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Customer Review

GT-2016 相关抗体

Top Publications Citing Use of Products

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

GT-2016 is a potent, selective, and brain penetrant histamine H3 receptor antagonist with a Ki of 43.8 nM. GT-2016 displays selectivity against H1 and H2 receptors, and has non-active against histamine methyltransferase[1].

IC50 & Target[1]

H3 Receptor

43.8 nM (Ki)

分子量

317.47

Formula

C19H31N3O
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

GT-2016 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

GT-2016152241-24-2GT2016GT 2016Histamine Receptorhistamine H3 receptorInhibitorinhibitorinhibit

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产品名称：
GT-2016
目录号：
HY-107559
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