1. GPCR/G Protein Neuronal Signaling
  2. Cannabinoid Receptor
  3. GW 833972A

GW 833972A 是一种选择性的 CB2 受体激动剂。GW 833972A 抑制受诱导神经去极化,并在动物模型中抑制柠檬酸引起的咳嗽。

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GW 833972A Chemical Structure

GW 833972A Chemical Structure

CAS No. : 1092502-33-4

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规格 价格 是否有货 数量
5 mg ¥4925
3 - 4 周
10 mg   询价  
50 mg   询价  

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Customer Review

查看 Cannabinoid Receptor 亚型特异性产品:

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

GW 833972A is a selective CB2 receptor agonist. GW 833972A inhibits induced nerve depolarization and citric acid-induced cough in animal models[1].

IC50 & Target[1]

hCB2-R

7.3 (pEC50)

rat CB2-R

7.5 (pEC50)

体外研究
(In Vitro)

GW 833972A (0.3-300 μM; 10 min) 抑制辣椒素诱导的人和豚鼠去极化,还抑制前列腺素 E(2) 和高渗盐水诱导的豚鼠离体迷走神经去极化[1]

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

体内研究
(In Vivo)

GW 833972A (30 mg/kg, 2 mL/kg;腹腔注射; 单次剂量, 试验开始前 30 min 注射) 能够抑制柠檬酸诱导的有意识豚鼠的咳嗽症状。它还抑制辣椒素引起的主支气管血浆蛋白渗出现象[1]

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

分子量

444.24

Formula

C18H14Cl2F3N5O

CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.

纯度 & 产品资料
参考文献
  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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产品名称:
GW 833972A
目录号:
HY-101765
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