2. Immunology/Inflammation
  3. PSMA
  4. PSMA-IN-1

PSMA-IN-1 (compound 23) 是 PSMA 的抑制剂，其 Ki 值为 2.49 nM。PSMA-IN-1 在 PSMA+ 荷瘤模型中以高选择性和特异性抑制肿瘤生长。PSMA-IN-1 也是一种用作肿瘤示踪的 NIR (λEX: 620 nm; λEM: 670 nm) 染料。PSMA-IN-1 可用于研究前列腺癌。

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PSMA-IN-1 Chemical Structure

PSMA-IN-1 Chemical Structure

1.  客户无需承担相应的运输费用。

2.  同一机构（单位）同一产品试用装仅限申领一次，同一机构（单位）一年内

     可免费申领三个不同产品的试用装。

3.  试用装只面向终端客户。

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PSMA-IN-1 相关抗体

Top Publications Citing Use of Products

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

PSMA-IN-1 (compound 23) is an inhibitor of PSMA with a Ki value of 2.49 nM. PSMA-IN-1 inhibits tumor growth with high selectivity and specificity in PSMA+ xenograft models. PSMA-IN-1 is a NIR probe (λEX: 620 nm; λEM: 670 nm) used for tumor disappearance. PSMA-IN-1 can be used for research on prostate cancer[1].

体内研究
(In Vivo)

PSMA-IN-1 (0.33 mg/kg, i.v., 一次) 是一种用作肿瘤示踪的 NIR (λEX: 620 nm; λEM: 670 nm) 染料，在注射后不同时间段获取图像 (2, 4, 8, 12, 24, and 48 h) [1]。
PSMA-IN-1 (0.33 mg/kg, i.v., 一次) 在 22Rv1 构建的BALB/C 裸鼠荷瘤模型中以高选择性和特异性抑制肿瘤生长[1]。

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model: 22Rv1 xenograft models in BALB/C nude mice[1]
Dosage: 0.33 mg/kg
Administration: Intravenous injection (i.v.), sacrificed at 55 h post-injection
Result: Increased TNR (tumor-to-normal tissue ratio) values from 3.20 at 2 h to 6.27 at 48 h.
分子量

1333.40

Formula

C66H80N10O20
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

PSMA-IN-1 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

PSMA-IN-1PSMAProstate-specific membrane antigen22Rv1selectivexenograftprostate cancerInhibitorinhibitorinhibit

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产品名称：
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目录号：
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