1. GPCR/G Protein Neuronal Signaling Immunology/Inflammation
  2. Histamine Receptor
  3. ROS 234

ROS 234 是有效的 H3 拮抗剂,对豚鼠回肠 H3 受体的pKB 值为 9.46,大鼠大脑的 pKi 值为 8.90,离体大鼠大脑皮层的 ED50 值为 19.12 mg/kg (腹腔注射)。ROS 234 具有较差的中枢通路。

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ROS 234 Chemical Structure

ROS 234 Chemical Structure

CAS No. : 184576-87-2

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Other Forms of ROS 234:

  • 生物活性

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  • 参考文献

生物活性

ROS 234 is a potent H3 antagonist, with a pKB of 9.46 for Guinea-pig ileum H3-receptor, a pKi of 8.90 for Rat cerebral cortex H3-receptor, and a ED50 of 19.12 mg/kg (ip) in ex vivo of Rat cerebral cortex. ROS 234 diaplays poor central access[1][2].

IC50 & Target[1]

rat H3 receptor

8.90 (pKi)

体内研究
(In Vivo)

ROS 234 centrally injected, significantly shortens pentobarbital narcosis[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

分子量

241.29

Formula

C13H15N5

CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.

纯度 & 产品资料
参考文献
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  • 稀释计算器

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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产品名称:
ROS 234
目录号:
HY-107563
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