1. Metabolic Enzyme/Protease Autophagy Apoptosis
  2. Dipeptidyl Peptidase Autophagy Ferroptosis
  3. Linagliptin-d4

Linagliptin-d4  (Synonyms: 利格列汀-d4; BI 1356-d4)

目录号: HY-10284S 纯度: 99.62%
COA 产品使用指南

Linagliptin-d4 是 Linagliptin 氘代物。Linagliptin 是一种有效,选择性的 DPP-4 抑制剂,IC50 值为 1 nM。

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Linagliptin-d<sub>4</sub> Chemical Structure

Linagliptin-d4 Chemical Structure

CAS No. : 2140263-92-7

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1 mg ¥4500
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查看 Dipeptidyl Peptidase 亚型特异性产品:

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

Linagliptin-d4 is deuterium labeled Linagliptin. Linagliptin is a highly potent, selective DPP-4 inhibitor with IC50 of 1 nM. Linagliptin-d4 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.

IC50 & Target

DPP-4

 

体外研究
(In Vitro)

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

分子量

476.57

Formula

C25H24D4N8O2

CAS 号
性状

固体

颜色

Off-white to light yellow

中文名称

利格列汀-d4;利拉利汀-d4;利格利汀-d4

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式
Powder -20°C 3 years
In solvent -80°C 6 months
-20°C 1 month
纯度 & 产品资料
参考文献
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  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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产品名称:
Linagliptin-d4
目录号:
HY-10284S
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