1. Others Membrane Transporter/Ion Channel Neuronal Signaling Autophagy
  2. Isotope-Labeled Compounds Calcium Channel Autophagy
  3. (R)-(-)-Felodipine-d5

(R)-(-)-Felodipine-d5 是 (R)-(-)-Felodipine 的氘代物。(R)-(-)-Felodipine 是 Felodipine 的异构体。Felodipine 是一种二氢吡啶,是一种有效的血管选择性钙通道 (b>calcium channel) 拮抗剂。Felodipine 通过选择性作用于血管平滑肌,尤其是阻力血管来降低血压。Felodipine 是具有抗高血压活性,可诱导自噬。Felodipine 可以跨越血脑屏障。

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(R)-(-)-Felodipine-d<sub>5</sub> Chemical Structure

(R)-(-)-Felodipine-d5 Chemical Structure

CAS No. : 1217744-87-0

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  • 生物活性

  • 纯度 & 产品资料

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生物活性

(R)-(-)-Felodipine-d5 is the deuterium labeled (R)-(-)-Felodipine. (R)-(-)-Felodipine is the S enantiomer of Felodipine. Felodipine, a dihydropyridine, is a potent, vasoselective calcium channel antagonist. Felodipine lowers blood pressure (BP) by selective action on vascular smooth muscle, especially in the resistance vessels. Felodipine, an anti-hypertensive agent, induces autophagy. Felodipine can cross the blood-brain barrier[1][2][3].

体外研究
(In Vitro)

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

分子量

389.28

Formula

C18H14D5Cl2NO4

CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.

纯度 & 产品资料
参考文献
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产品名称:
(R)-(-)-Felodipine-d5
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