1. Others GPCR/G Protein Neuronal Signaling Immunology/Inflammation
  2. Isotope-Labeled Compounds Histamine Receptor
  3. Bilastine-d6

Bilastine-d6  (Synonyms: 比拉斯汀 d6)

目录号: HY-14447S
产品使用指南

Bilastine-d6 是 Bilastine 的氘代物。Bilastine是组胺H1受体拮抗剂,可作用于变应性鼻结膜炎和荨麻疹。

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Bilastine-d<sub>6</sub> Chemical Structure

Bilastine-d6 Chemical Structure

CAS No. : 1215358-58-9

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     可免费申领三个不同产品的试用装。

3.  试用装只面向终端客户

规格 价格 是否有货 数量
1 mg ¥5700
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Top Publications Citing Use of Products
  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

Bilastine-d6 is the deuterium labeled Bilastine. Bilastine is a selective histamine H1 receptor antagonist used for treatment of allergic rhinoconjunctivitis and urticaria[1][2].

IC50 & Target

H1 Receptor

 

体外研究
(In Vitro)

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

分子量

469.65

Formula

C28H31D6N3O3

CAS 号
中文名称

比拉斯汀 d6

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.

溶解性数据
In Vitro: 

DMSO 中的溶解度 : 10 mg/mL (21.29 mM; 超声加热助溶; 吸湿的 DMSO 对产品的溶解度有显著影响,请使用新开封的 DMSO)

配制储备液
浓度 溶剂体积 质量 1 mg 5 mg 10 mg
1 mM 2.1292 mL 10.6462 mL 21.2925 mL
5 mM 0.4258 mL 2.1292 mL 4.2585 mL
查看完整储备液配制表
  • 摩尔计算器

  • 稀释计算器

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量
=
浓度
×
体积
×
分子量 *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start)

C1

×
体积 (start)

V1

=
浓度 (final)

C2

×
体积 (final)

V2

动物溶解方案计算器
请输入动物实验的基本信息:

给药剂量

mg/kg

动物的平均体重

g

每只动物的给药体积

μL

动物数量

由于实验过程有损耗,建议您多配一只动物的量
计算结果
工作液所需浓度 : mg/mL
纯度 & 产品资料
参考文献

完整储备液配制表

可选溶剂 浓度 溶剂体积 质量 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 2.1292 mL 10.6462 mL 21.2925 mL 53.2311 mL
5 mM 0.4258 mL 2.1292 mL 4.2585 mL 10.6462 mL
10 mM 0.2129 mL 1.0646 mL 2.1292 mL 5.3231 mL
15 mM 0.1419 mL 0.7097 mL 1.4195 mL 3.5487 mL
20 mM 0.1065 mL 0.5323 mL 1.0646 mL 2.6616 mL
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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产品名称:
Bilastine-d6
目录号:
HY-14447S
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