2. GPCR/G Protein
  3. Adenosine Receptor
  4. BW-534U87

BW-534U87 是一种口服有效的腺苷 A1 受体 (adenosine A1 receptor) 激动剂以及竞争性的腺苷脱氨酶 (ADA) 抑制剂 (Ki=7 μM)。BW-534U87 能提高大脑中的腺苷水平，并抑制癫痫样活动。BW-534U87 在动物癫痫模型中显示出抗惊厥效果。BW-534U87 有望用于癫痫及腺苷相关神经精神障碍的研究。

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BW-534U87

BW-534U87 Chemical Structure

CAS No. : 143153-93-9

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BW-534U87 相关抗体

Top Publications Citing Use of Products

查看 Adenosine Receptor 亚型特异性产品:

查看所有亚型
Adenosine A1 receptor (A1R) Adenosine A2A receptor (A2AR) Adenosine A2B receptor (A2BR) Adenosine A3 receptor (A3R)

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

BW-534U87 is an orally active adenosine A1 receptor agonist and competitive adenosine deaminase (ADA) inhibitor (Ki=7 μM). BW-534U87 elevates brain adenosine levels and suppresses epileptiform activity. BW-534U87 demonstrate anticonvulsant efficacy in animal seizure models. BW-534U87 is promising for research of epilepsy and adenosine-related neuropsychiatric disorders[1].

IC50 & Target

A1AR

 

分子量

297.69

Formula

C12H10ClF2N5
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

BW-534U87 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

BW-534U87143153-93-9Adenosine ReceptorP1 receptoradenosine A1 receptorADAneuropsychiatric disordersInhibitorinhibitorinhibit

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产品名称：
BW-534U87
目录号：
HY-19130
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