2. GPCR/G Protein Neuronal Signaling Metabolic Enzyme/Protease
  3. Cannabinoid Receptor FAAH
  4. CB2R/FAAH modulator-1

CB2R/FAAH modulator-1 是一种大麻素 2 型受体 (CB2R) 完全激动剂，对 CB2R 和 CB1R 的 Ki 分别为 14.8 nM 和 241.3 nM。CB2R/FAAH modulator-1 是一种脂肪酸酰胺水解酶 (FAAH) 抑制剂，IC50 为 4 μM。CB2R/FAAH modulator-1 减少促炎并增加抗炎细胞因子的产生。

MCE 的所有产品仅用作科学研究或药证申报，我们不为任何个人用途提供产品和服务

CB2R/FAAH modulator-1 Chemical Structure

CB2R/FAAH modulator-1 Chemical Structure

CAS No. : 928892-60-8

1.  客户无需承担相应的运输费用。

2.  同一机构（单位）同一产品试用装仅限申领一次，同一机构（单位）一年内

     可免费申领三个不同产品的试用装。

3.  试用装只面向终端客户。

规格 是否有货
50 mg   询价  
100 mg   询价  
250 mg   询价  

* Please select Quantity before adding items.

Customer Review

CB2R/FAAH modulator-1 相关抗体

Top Publications Citing Use of Products

查看 Cannabinoid Receptor 亚型特异性产品:

查看所有亚型
CB1 CB2

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

CB2R/FAAH modulator-1 is a cannabinoid type 2 receptor (CB2R) full agonist with Kis of 14.8 nM and 241.3 nM for CB2R and CB1R, respectively. CB2R/FAAH modulator-1 is a fatty acid amide hydrolase (FAAH) inhibitor with an IC50 of 4 μM. CB2R/FAAH modulator-1 decreases pro-inflammatory and increases anti-inflammatory cytokines production[1].

IC50 & Target[1]

CB2R

14.8 nM (Ki)

CB2R

123.6 nM (EC50)

CB1R

241.3 nM (Ki)

CB1R

489 nM (EC50)

体外研究
(In Vitro)

CB2R/FAAH modulator-1 (化合物 13; 10 μM; 24 小时) 减少未刺激的单核细胞和巨噬细胞中促炎细胞因子 TNFα、IFN-γ、IL-1β 和 IL6 的产生[1] .

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

CB2R/FAAH modulator-1 相关抗体:
分子量

361.48

Formula

C24H27NO2
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

CB2R/FAAH modulator-1 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

CB2R/FAAH modulator-1928892-60-8Cannabinoid ReceptorFAAHFatty acid amide hydrolasecannabinoid type 2 receptorCB2RCB1Rfatty acid amide hydrolaseanti-inflammatory cytokinesTNFαIFN-γIL-1βIL6Inhibitorinhibitorinhibit

您最近查看的产品:

Your information is safe with us. * Required Fields.

   产品名称：

  

* 需求量：

* 客户姓名：

 

* Email：

* 电话：

 

* 公司或机构名称：

   留言给我们：

Bulk Inquiry

Inquiry Information

产品名称：
CB2R/FAAH modulator-1
目录号：
HY-152251
需求量：

Request for HNMR Report

Please fill out this form to request the QC report. We will send it to your Email address shortly.

Your information is safe with us. * Required Fields.

   产品名称：

  

* Lot #：

* 客户姓名：

 

* Email：

   电话：

 

* 部门：

* 公司或机构名称：

 

   留言给我们：

Request for HNMR Report

We have received your request and will respond to you as soon as possible.

嗨！很高兴为您提供帮助！

尊敬的 MCE 客户您好，
请您选择所在区域，我们将转接对应客服为您服务！

热门区域

A

B

C

F

G

H

J

L

N

Q

S

T

X

Y

Z

热 A B C F G H J L N Q S T X Y Z