1. Antibody-drug Conjugate/ADC Related
  2. Drug-Linker Conjugates for ADC
  3. MC-Gly-Gly-Phe-Gly-Cyclobutanecarboxylic-Exatecan

MC-Gly-Gly-Phe-Gly-Cyclobutanecarboxylic-Exatecan 

目录号: HY-147307 纯度: 98.66%
COA 产品使用指南

MC-Gly-Gly-Phe-Gly-Cyclobutanecarboxylic-Exatecan 是抗体偶联活性分子 ADC 的一部分,由 ADC linker (MC-Gly-Gly-Phe-Gly-Cyclobutanecarboxylic) 和 DNA 拓扑异构酶 I (topoisomerase I) 抑制剂 Exatecan (HY-13631) 偶联而成。MC-Gly-Gly-Phe-Gly-Cyclobutanecarboxylic-Exatecan 合成的 ADC 可用于癌症的研究。

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MC-Gly-Gly-Phe-Gly-Cyclobutanecarboxylic-Exatecan Chemical Structure

MC-Gly-Gly-Phe-Gly-Cyclobutanecarboxylic-Exatecan Chemical Structure

CAS No. : 2414393-22-7

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1 mg ¥4500
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  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

MC-Gly-Gly-Phe-Gly-Cyclobutanecarboxylic-Exatecan is a agent-linker conjugate for ADC, contains the ADC linker (MC-Gly-Gly-Phe-Gly-Cyclobutanecarboxylic acid) and a DNA topoisomerase I inhibitor Exatecan (HY-13631). MC-Gly-Gly-Phe-Gly-Cyclobutanecarboxylic-Exatecan synthesized ADC can be used in study of cancer[1].

IC50 & Target

Camptothecins

 

分子量

1074.12

Formula

C55H60FN9O13

CAS 号
性状

固体

颜色

Off-white to light yellow

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

-20°C, sealed storage, away from moisture and light

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)

纯度 & 产品资料

纯度: 98.66%

参考文献

MC-Gly-Gly-Phe-Gly-Cyclobutanecarboxylic-Exatecan 相关分类

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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产品名称:
MC-Gly-Gly-Phe-Gly-Cyclobutanecarboxylic-Exatecan
目录号:
HY-147307
需求量: