1. Signaling Pathways
  2. Epigenetics
    PI3K/Akt/mTOR
  3. AMPK
  4. AMPK Inhibitors

AMPK Inhibitors

NUAK1

NUAK2

AMPK

AMPK α1β1γ1

AMPK α2β1γ1

AMPK α1β2γ1

AMPK α2β2γ1

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

AMPK Inhibitors & Activators
Product Name NUAK1 NUAK2 AMPK AMPK α1β1γ1 AMPK α2β1γ1 AMPK α1β2γ1 AMPK α2β2γ1 Purity
Dorsomorphin    
AMPK, Ki: 109 nM
        99.91%
Metformin    
AMPK
        99.98%
AICAR    
AMPK
        99.97%
Dorsomorphin dihydrochloride    
AMPK, Ki: 109 nM
        99.91%
Metformin hydrochloride    
AMPK
        99.92%
A-769662    
AMPK, EC50: 0.8 μM
        99.20%
MK8722    
AMPK
        99.37%
Bempedoic acid    
AMPK
        98.99%
AICAR phosphate    
AMPK
        99.80%
[6]-Gingerol    
AMPK
        99.45%
Phenformin hydrochloride    
AMPK
        99.29%
PF-06409577      
AMPK α1β1γ1, EC50: 7 nM
      99.44%
WZ4003
NUAK1, IC50: 20 nM
NUAK2, IC50: 100 nM
          98.88%
HTH-01-015
NUAK1, IC50: 100 nM
            98.81%
EX229      
AMPK α1β1γ1, Kd: 0.06 μM
AMPK α2β1γ1, Kd: 0.06 μM
AMPK α1β2γ1, Kd: 0.51 μM
  98.45%
Palmitelaidic Acid    
AMPK
        ≥99.0%
Narazaciclib
ARK5, IC50: 5 nM
            99.34%
Danthron    
AMPK
        99.19%
MRT199665
NUAK1, IC50: 3 nM
NUAK2, IC50: 120 nM
          99.92%
MOTS-c(human) acetate    
AMPK
        98.97%
ASP4132    
AMPK, EC50: 18 nM
        99.32%
MK-3903    
AMPK, EC50: 8 nM
        98.03%
RSVA405    
AMPK, EC50: 1 μM (in cell-based assays)
        99.58%
Metformin-d6 hydrochloride    
AMPK
        98.79%
Ginkgolide C    
AMPK
        ≥98.0%
MT 63-78    
AMPK, EC50: 25 μM
        98.50%
ZLN024 hydrochloride      
AMPK α1β1γ1, EC50: 0.42 μM
AMPK α2β1γ1, EC50: 0.95 μM
 
AMPK α2β2γ1, EC50: 0.13 μM
98.47%
Ampkinone    
AMPK
        99.28%
PF-06685249      
AMPK α1β1γ1, EC50: 12 nM
      98.32%
Gomisin J    
AMPK
        99.84%
SAMS    
AMPK
        99.88%
YLF-466D    
AMPK
        98.41%
PF-739      
AMPK α1β1γ1, EC50: 8.99 nM
AMPK α2β1γ1, EC50: 5.23 nM
AMPK α1β2γ1, EC50: 126 nM
AMPK α2β2γ1, EC50: 42.2 nM
98.05%
8-Chloroadenosine    
AMPK
        99.97%
3α-Hydroxymogrol    
AMPK
        99.88%
AMPK activator 1    
AMPK, EC50: 0.1 μM
        98.53%
IQZ23    
AMPK
       
PF-06679142      
AMPK α1β1γ1, EC50: 22 nM
     
Kazinol B    
AMPK
       
AMPK activator 8      
AMPK α1β1γ1, EC50: 11 nM
AMPK α2β1γ1, EC50: 27 nM
AMPK α1β2γ1, EC50: 4 nM
AMPK α2β2γ1, EC50: 2 nM
LRRK2-IN-8
NUAK1, IC50: 10-100 nM
           
Tanshinol borneol ester    
AMPK
       
AMPK activator 10    
AMPK
       
AMPK activator 2    
AMPK
       
Etilefrine    
AMPK
       
AMPK-IN-1            
AMPK α2β2γ1, EC50: 551 nM
LRRK2/NUAK1/TYK2-IN-1
NUAK1
           
AMPK activator 9        
AMPK α2β1γ1, EC50: 1.1 μM
   
AMPK activator 2 hydrochloride    
AMPK
        99.65%
ZLN024      
AMPK α1β1γ1, EC50: 0.42 μM
AMPK α2β1γ1, EC50: 0.95 μM
 
AMPK α2β2γ1, EC50: 0.13 μM