1. Signaling Pathways
  2. Epigenetics
    PI3K/Akt/mTOR
  3. AMPK
  4. AMPK Inhibitors

AMPK Inhibitors

NUAK1

NUAK2

AMPK

AMPK α1β1γ1

AMPK α2β1γ1

AMPK α1β2γ1

AMPK α2β2γ1

BRSK1

BRSK2

HUNK

AMPKα

Your Search Returned No Results.

Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

AMPK Inhibitors, Agonists & Activators
Product Name NUAK1 NUAK2 AMPK AMPK α1β1γ1 AMPK α2β1γ1 AMPK α1β2γ1 AMPK α2β2γ1 BRSK1 BRSK2 HUNK AMPKα Purity
Dorsomorphin    
AMPK, Ki: 109 nM
                99.91%
Metformin    
AMPK
                99.98%
AICAR    
AMPK
                99.98%
Dorsomorphin dihydrochloride    
AMPK, Ki: 109 nM
                99.91%
HDAC11-IN-2      
AMPK α1β1γ1
              99.52%
Metformin hydrochloride    
AMPK
                99.98%
A-769662    
AMPK, EC50: 0.8 μM
                99.33%
MK8722    
AMPK
                99.82%
Bempedoic acid    
AMPK
                99.97%
[6]-Gingerol    
AMPK
                99.68%
AICAR phosphate    
AMPK
                99.98%
Phenformin hydrochloride    
AMPK
                99.64%
EX229      
AMPK α1β1γ1, Kd: 0.06 μM
AMPK α2β1γ1, Kd: 0.06 μM
AMPK α1β2γ1, Kd: 0.51 μM
          99.44%
Palmitelaidic Acid    
AMPK
                99.4%
HTH-01-015
NUAK1, IC50: 100 nM
                    98.81%
WZ4003
NUAK1, IC50: 20 nM
NUAK2, IC50: 100 nM
                  98.03%
PF-06409577      
AMPK α1β1γ1, EC50: 7 nM
              99.83%
PF-739      
AMPK α1β1γ1, EC50: 8.99 nM
AMPK α2β1γ1, EC50: 5.23 nM
AMPK α1β2γ1, EC50: 126 nM
AMPK α2β2γ1, EC50: 42.2 nM
        99.79%
Danthron    
AMPK
                99.41%
MOTS-c(human) acetate    
AMPK
                98.97%
MRT199665
NUAK1, IC50: 3 nM
NUAK2, IC50: 120 nM
                  99.74%
Narazaciclib
ARK5, IC50: 5 nM
                    98.66%
Ginkgolide C    
AMPK
                ≥98.0%
Metformin-d6 hydrochloride    
AMPK
                99.98%
ASP4132    
AMPK, EC50: 18 nM
                99.32%
RSVA405    
AMPK, EC50: 1 μM (in cell-based assays)
                99.72%
ZLN024 hydrochloride      
AMPK α1β1γ1, EC50: 0.42 μM
AMPK α2β1γ1, EC50: 0.95 μM
 
AMPK α2β2γ1, EC50: 0.13 μM
        98.51%
8-Chloroadenosine    
AMPK
                99.97%
MOTS-c (human)    
AMPK
                99.90%
MT 63-78    
AMPK, EC50: 25 μM
                98.00%
SAMS    
AMPK
                99.88%
A17                    
AMPKα1
99.4%
MK-3903    
AMPK, EC50: 8 nM
                98.03%
PF-06685249      
AMPK α1β1γ1, EC50: 12 nM
              98.00%
Ampkinone    
AMPK
                99.28%
YLF-466D    
AMPK
                99.02%
Myricanol    
AMPK
                ≥98.0%
Gomisin J    
AMPK
                99.87%
AMPK activator 2 hydrochloride    
AMPK
                99.65%
Etilefrine    
AMPK
               
AMPK activator 1    
AMPK, EC50: 0.1 μM
                98.53%
3α-Hydroxymogrol    
AMPK
                99.88%
AMPK-IN-1            
AMPK α2β2γ1, EC50: 551 nM
       
IQZ23    
AMPK
               
PF-06679142      
AMPK α1β1γ1, EC50: 22 nM
             
HUNK Human Pre-designed siRNA Set A                  
HUNK
 
Kazinol B    
AMPK
               
AMPK activator 8      
AMPK α1β1γ1, EC50: 11 nM
AMPK α2β1γ1, EC50: 27 nM
AMPK α1β2γ1, EC50: 4 nM
AMPK α2β2γ1, EC50: 2 nM
       
LRRK2-IN-8
NUAK1, IC50: 10-100 nM
                   
Tanshinol borneol ester    
AMPK
               
AMPK activator 10    
AMPK
               
AMPK activator 2    
AMPK
               
BRSK1 Human Pre-designed siRNA Set A              
BRSK1
     
AMPK-IN-6    
AMPK, IC50: 0.093 μM
               
LRRK2/NUAK1/TYK2-IN-1
NUAK1
                   
AMPK activator 9        
AMPK α2β1γ1, EC50: 1.1 μM
           
Brsk2 Rat Pre-designed siRNA Set A                
BRSK2
   
ZLN024      
AMPK α1β1γ1, EC50: 0.42 μM
AMPK α2β1γ1, EC50: 0.95 μM
 
AMPK α2β2γ1, EC50: 0.13 μM