DYRK Inhibitors

DYRK1

DYRK2

DYRK3

DYRK4

HIPK

PRP4

DYRK Inhibitors

Product Name	DYRK1	DYRK2	DYRK3	DYRK4	HIPK	PRP4	Purity
Harmine	DYRK1A						99.97%
AZ191	DYRK1B						99.98%
GSK-626616	DYRK1	DYRK2	DYRK3				99.77%
GNF2133	DYRK1A, IC₅₀: 0.0062 μM						98.12%
GSK3-IN-10	DYRK1A, IC₅₀: 170 nM DYRK1B, IC₅₀: 47 nM	DYRK2, IC₅₀: 800 nM
KTD-092	DYRK1A, IC₅₀: 22 nM
Dyrk1A-IN-13	DYRK1A, IC₅₀: 41 nM DYRK1B, IC₅₀: 78 nM
T025	DYRK1A, Kd: 0.074 nM DYRK1B, Kd: 1.5 nM	DYRK2, Kd: 32 nM					99.64%
DYRK1-IN-1	DYRK1A, IC₅₀: 220 nM DYRK1A, Kd: 3 nM DYRK1B, Kd: 56 nM						99.71%
GNF4877	DYRK1A, IC₅₀: 6 nM						99.82%
Harmine hydrochloride	DYRK1A						99.98%
Protein kinase inhibitor 1 hydrochloride	DYRK1	DYRK2					≥98.0%
INDY	DYRK1A DYRK1B						99.32%
EHT 1610	DYRK1A DYRK1B						98.16%
ILK-IN-3	DYRK1						99.62%
RO5454948	DYRK1A, IC₅₀: 22 nM DYRK1B, IC₅₀: 68 nM						99.53%
ML167	DYRK1A, IC₅₀: ＞10000 nM DYRK1B, IC₅₀: 4420 nM						98.62%
Dyrk1A-IN-5	DYRK1A, IC₅₀: 6 nM DYRK1B, IC₅₀: 600 nM	DYRK2, IC₅₀: >10000 nM					98.56%
AZ-Dyrk1B-33	DYRK1B						99.95%
LDN-192960	DYRK1	DYRK2					99.58%
EHT 5372	DYRK1A, IC₅₀: 0.22 nM DYRK1B, IC₅₀: 0.28 nM	DYRK2, IC₅₀: 10.8 nM		DYRK4, IC₅₀: 93.2 nM			98.12%
Dyrk1A-IN-4	DYRK1A, IC₅₀: 2 nM	DYRK2, IC₅₀: 6 nM					99.90%
CLK1-IN-3	DYRK1A, IC₅₀: 1521 nM						98.54%
ON 108600	DYRK1A, IC₅₀: 0.016 μM DYRK1B, IC₅₀: 0.007 μM	DYRK2, IC₅₀: 0.028 μM					99.73%
LDN-209929 dihydrochloride		DYRK2					98.33%
YK-2-69		DYRK2, IC₅₀: 9 nM					99.57%
7-Deazaguanine	DYRK1A						≥99.0%
HTH-01-091				DYRK4, IC₅₀: 41.8 nM			98.64%
DYRKs-IN-1 hydrochloride	DYRK1A, IC₅₀: 5 nM DYRK1B, IC₅₀: 8 nM						99.71%
LDN-192960 hydrochloride	DYRK1	DYRK2					99.78%
KH-CB20	DYRK1A, IC₅₀: 57.8 nM						99.80%
MU1210		DYRK2, IC₅₀: 1309 nM					99.50%
(R)-(+)-O-Demethylbuchenavianine	DYRK1A						98.67%
DYRKs-IN-1	DYRK1A, IC₅₀: 5 nM DYRK1B, IC₅₀: 8 nM
GNF2133 hydrochloride	DYRK1A, IC₅₀: 0.0062 μM
MBM-55S	DYRK1A, IC₅₀: 6.5 nM
Dyrk1A/α-synuclein-IN-2	DYRK1A
Haspin-IN-2	DYRK1A, IC₅₀: 917 nM
Dyrk1A-IN-7	DYRK1A, IC₅₀: 28 nM
Dyrk1A-IN-8	DYRK1A, IC₅₀: 209 nM
Dyrk1A/B-IN-1	DYRK1A, Ki: 67.8 nM DYRK1B, Ki: 237.9 nM
Haspin-IN-1	DYRK1A, IC₅₀: 916.3 nM
Dyrk1A-IN-1	DYRK1
JH-XVII-10	DYRK1A, IC₅₀: 3 nM DYRK1B, IC₅₀: 5 nM
hAChE-IN-8	DYRK1A, IC₅₀: >10 μM
JH-XIV-68-3	DYRK1
ZJCK-6-46	DYRK1A, IC₅₀: 0.68 nM DYRK1B, IC₅₀: 1.02 nM	DYRK2, IC₅₀: 14.18 nM	DYRK3, IC₅₀: 17.48 nM	DYRK4, IC₅₀: 401.3 nM
Dyrk1A/α-synuclein-IN-1	DYRK1A, IC₅₀: 177 nM
Cnksr3 Rat Pre-designed siRNA Set A						PRP4
Hipk2 Rat Pre-designed siRNA Set A					HIPK1
Norharmine	DYRK1A
Dyrk1A-IN-2	DYRK1A, EC₅₀: 37 nM
Dyrk1A-IN-11	DYRK1A, EC₅₀: 0.0021 μM
Dyrk1A-IN-12	DYRK1A, IC₅₀: 95 nM
RD0392	DYRK1A

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