1. GPCR/G Protein
    Neuronal Signaling
  2. Opioid Receptor
  3. DPI-3290

DPI-3290 (Synonyms: Org 41793)

目录号: HY-19231
产品使用指南

DPI-3290 (Org 41793) 是一种有效的,特异性的阿片受体 (opioid receptors) 激动剂,对 δ-,μ- 和 κ- 阿片受体的 Ki 值分别为 0.18 nM,0.46 nM 和 0.62 nM。DPI-3290 是一系列新型中枢作用药物之一,具有强烈的抗伤害作用。

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DPI-3290 Chemical Structure

DPI-3290 Chemical Structure

CAS No. : 182417-73-8

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Description

DPI-3290 (Org 41793) is a potent and specific opioid receptors agonist with Ki values of 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively。DPI-3290 is one of a series of novel centrally acting agents with potent antinociceptive activity[1].

IC50 & Target

IC50: 0.18 nM (δ-opioid receptor), 0.46 nM (μ-opioid receptor) and 0.62 nM (κ-opioid receptor)[1]

In Vivo

DPI-3290 (Org 41793) (intravenous; 0.05 mg/kg) produces a 50% antinociceptive response in rats[1].

Molecular Weight

487.61

Formula

C₃₀H₃₄FN₃O₂

CAS No.

182417-73-8

SMILES

O=C(N(C1=CC=CC(F)=C1)C)C2=CC=CC([C@@H](N3[C@@H](C)CN(CC=C)[C@H](C)C3)C4=CC=CC(O)=C4)=C2

Shipping

Room temperature in continental US; may vary elsewhere

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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产品名称:
DPI-3290
目录号:
HY-19231
需求量:

DPI-3290

Cat. No.: HY-19231