2. GPCR/G Protein
  3. Leukotriene Receptor
  4. MEN-91507

MEN-91507 是一种具有口服活性的半胱氨酰白三烯受体 1 (CysLTR1) 受体拮抗剂。MEN-91507 表现出对 Leukotriene D4 (HY-113456) 诱导的钙瞬变的不可逆拮抗作用，其 pKb 值为 10.25。MEN-91507 能抑制 Leukotriene D4 诱导的豚鼠支气管收缩和微血管渗漏。MEN-91507 可用于炎症、免疫学研究。

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MEN-91507

MEN-91507 Chemical Structure

CAS No. : 197506-04-0

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MEN-91507 相关抗体

Top Publications Citing Use of Products

查看 Leukotriene Receptor 亚型特异性产品:

查看所有亚型
LTB4 LTC4/CysLT2 LTD4/CysLT1 LTE4

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

MEN-91507 is an orally activecysteinyl leukotriene receptor 1 (CysLTR1) receptor antagonist. MEN-91507 behaves as insurmountable antagonist of Leukotriene D4 (HY-113456)-induced calcium transients, with a pKb of 10.25. MEN-91507 can inhibit Leukotriene D4-induced bronchoconstriction and microvascular leakage in guinea-pigs. MEN-91507 can be used for the researches of inflammation, immunology[1].

IC50 & Target[1]

CysLT1

 

分子量

482.51

Formula

C28H23FN4O3
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

MEN-91507 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

MEN-91507197506-04-0MEN91507MEN 91507Leukotriene Receptorleukotriene receptorCysLTR1Leukotriene D4bronchoconstrictionmicrovascular leakageguinea-pigInhibitorinhibitorinhibit

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产品名称：
MEN-91507
目录号：
HY-19395
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