1. PROTAC
  2. E3 Ligase Ligand-Linker Conjugate
  3. (S,R,S)-AHPC-Me-C5-COOH

(S,R,S)-AHPC-Me-C5-COOH 

目录号: HY-130849
产品使用指南

(S,R,S)-AHPC-Me-C5-COOH 是一种合成的 E3 连接酶配体结合物,它结合了 VHL 配体和连接子。(S,R,S)-AHPC-Me-C5-COOH 可用于 PROTAC DT2216 (HY-130604)。

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(S,R,S)-AHPC-Me-C5-COOH Chemical Structure

(S,R,S)-AHPC-Me-C5-COOH Chemical Structure

CAS No. : 2229976-21-8

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Description

(S,R,S)-AHPC-Me-C5-COOH is a synthesized E3 ligase ligand-linker conjugate that incorporates the a VHL ligand and a linker. (S,R,S)-AHPC-Me-C5-COOH can be used in PROTAC DT2216 (HY-130604)[1].

IC50 & Target[1]

VHL

 

In Vitro

DT2216 is a selective B-cell lymphoma extra large (BCL-XL) PROTAC degrader[1].

Molecular Weight

586.74

Formula

C₃₀H₄₂N₄O₆S

CAS No.

2229976-21-8

SMILES

O=C(N[C@H](C1=CC=C(C2=C(C)N=CS2)C=C1)C)[C@H]3N(C([C@H](C(C)(C)C)NC(CCCCCC(O)=O)=O)=O)C[C@H](O)C3

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Keywords:

(S,R,S)-AHPC-Me-C5-COOHE3 Ligase Ligand-Linker ConjugateInhibitorinhibitorinhibit

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产品名称:
(S,R,S)-AHPC-Me-C5-COOH
目录号:
HY-130849
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